SYNTHESIS VIA A CYCLIC DIOXATRICHLOROPHOSPHORANE OF 1,3-DIBENZYL-2-PHOSPHONOOXY CITRATE

被引：9

作者：

PANKOWSKI, AH ^{[1
]}

MEEHAN, JD ^{[1
]}

SALLIS, JD ^{[1
]}

机构：

[1] UNIV TASMANIA,DEPT BIOCHEM,HOBART,TAS 7001,AUSTRALIA

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(00)76002-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Phosphorylation of tribenzyl citrate with PCl5 proceeds via a cyclic dioxatrichlorophosphorane and results in the formation of 1,3-dibenzyl-2-phosphonooxy citrate. A mechanism for the phosphorylation and ester hydrolysis is proposed and the usefulness of the diester for producing triesters is discussed.

引用

页码：927 / 930

页数：4

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