SYNTHESIS OF C-3 HALOGEN-SUBSTITUTED APOCODEINES AND APOMORPHINES

被引：15

作者：

SIMON, C

HOSZTAFI, S

MAKLEIT, S ^{[1
]}

BERENYI, S

机构：

[1] LAJOS KOSSUTH UNIV, DEPT ORGAN CHEM, POB 20, H-4010 DEBRECEN, HUNGARY

[2] ALKALOIDA CHEM FACTORY, H-4440 TISZAVASVARI, HUNGARY

来源：

SYNTHETIC COMMUNICATIONS | 1991年 / 21卷 / 22期

关键词：

D O I：

10.1080/00397919108021590

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new effective method has been elaborated for the preparation of the hitherto unknown C-3 halogene derivatives (Cl, Br) of apocodeine and apomorphine, as well as of their N-demethyl-N-substituted (N-propyl, N-alkyl) analogues. These compounds are expected to possess an effect on the dopamine receptor system.

引用

页码：2309 / 2316

页数：8

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