THE CALCIUM ANTAGONISTIC EFFECTS OF CYPROHEPTADINE ON CONTRACTION, MEMBRANE ELECTRICAL EVENTS AND CALCIUM INFLUX IN THE GUINEA-PIG TAENIA-COLI

被引:43
作者
LOWE, DA [1 ]
MATTHEWS, EK [1 ]
RICHARDSON, BP [1 ]
机构
[1] UNIV CAMBRIDGE, DEPT PHARMACOL, CAMBRIDGE, ENGLAND
关键词
SMOOTH-MUSCLE; MECHANICAL-ACTIVITY; POTASSIUM; LANTHANUM; INSULIN; TENSION; SODIUM; DRUGS;
D O I
10.1111/j.1476-5381.1981.tb10476.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:651 / 663
页数:13
相关论文
共 29 条
[1]   INOTROPIC AND ELECTROPHYSIOLOGICAL ACTIONS OF VERAPAMIL AND D-600 IN MAMMALIAN MYOCARDIUM .1. PATTERN OF INOTROPIC EFFECTS OF RACEMIC COMPOUNDS [J].
BAYER, R ;
HENNEKES, R ;
KAUFMANN, R ;
MANNHOLD, R .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1975, 290 (01) :49-68
[2]   SUCROSE-GAP TECHNIQUE WITH PRESSED RUBBER MEMBRANES [J].
BOEV, K ;
GOLENHOFEN, K .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1974, 349 (03) :277-283
[3]   MECHANISMS OF ACTION OF TRANSMITTERS AND OTHER SUBSTANCES ON SMOOTH-MUSCLE [J].
BOLTON, TB .
PHYSIOLOGICAL REVIEWS, 1979, 59 (03) :606-718
[4]   USE OF LANTHANUM TO ESTIMATE NUMBERS OF EXTRACELLULAR CATION-EXCHANGING SITES IN GUINEA-PIGS TAENIA-COLI, AND ITS EFFECTS ON TRANSMEMBRANE MONOVALENT ION MOVEMENTS [J].
BRADING, AF ;
WIDDICOMBE, JH .
JOURNAL OF PHYSIOLOGY-LONDON, 1977, 266 (02) :255-273
[5]  
BULBRING E, 1954, J PHYSIOL-LONDON, V125, P302
[6]   MECHANISM BY WHICH CYPROHEPTADINE INHIBITS INSULIN-SECRETION [J].
DONATSCH, P ;
LOWE, DA ;
RICHARDSON, BP ;
TAYLOR, P .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 70 (03) :355-362
[7]   EFFECT OF POTASSIUM ON MECHANICAL-ACTIVITY OF TAENIA-COLI, UTERUS AND PORTAL-VEIN OF GUINEA-PIG [J].
GABELLA, G .
QUARTERLY JOURNAL OF EXPERIMENTAL PHYSIOLOGY AND COGNATE MEDICAL SCIENCES, 1978, 63 (02) :125-146
[8]   SELECTIVE SUPPRESSION OF SOME COMPONENTS OF SPONTANEOUS ACTIVITY IN VARIOUS TYPES OF SMOOTH MUSCLE BY IPROVERATRIL (VERAPAMIL) [J].
GOLENHOFEN, K ;
LAMMEL, E .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1972, 331 (03) :233-+