EVIDENCE OF THE PREFERENTIAL INVOLVEMENT OF MU-RECEPTORS IN ANALGESIA USING ENKEPHALINS HIGHLY SELECTIVE FOR PERIPHERAL MU-RECEPTOR OR DELTA-RECEPTOR

被引：72

作者：

GACEL, G ^{[1
]}

FOURNIEZALUSKI, MC ^{[1
]}

FELLION, E ^{[1
]}

ROQUES, BP ^{[1
]}

机构：

[1] FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 10期

关键词：

D O I：

10.1021/jm00142a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1119 / 1124

页数：6

共 46 条

[1]

BAXTER MG, 1977, P BRIT PHARMACOL SOC, pP455

[2] STRUCTURAL REQUIREMENTS FOR OPIOID ACTIVITY OF ANALOGS OF ENKEPHALINS [J].

BEDDELL, CR ;

CLARK, RB ;

HARDY, GW ;

LOWE, LA ;

UBATUBA, FB ;

VANE, JR ;

WILKINSON, S ;

CHANG, KJ ;

CUATRECASAS, P ;

MILLER, RJ .

PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1977, 198 (1132) :249-265

[3] OPIATE RECEPTOR AFFINITIES AND BEHAVIORAL-EFFECTS OF ENKEPHALIN - STRUCTURE-ACTIVITY RELATIONSHIP OF 10 SYNTHETIC PEPTIDE ANALOGS [J].

CHANG, JK ;

FONG, BTW ;

PERT, A ;

PERT, CB .

LIFE SCIENCES, 1976, 18 (12) :1473-1481

[4] POSSIBLE ROLE OF DISTINCT MORPHINE AND ENKEPHALIN RECEPTORS IN MEDIATING ACTIONS OF BENZOMORPHAN DRUGS (PUTATIVE-KAPPA AND SIGMA-AGONISTS) [J].

CHANG, KJ ;

HAZUM, E ;

CUATRECASAS, P .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (08) :4469-4473

[5]

CHANG KJ, 1979, J BIOL CHEM, V254, P2160

[6]

CHESSELET MF, NATURE LONDON

[7] OPIATE RECEPTOR-BINDING AFFECTED DIFFERENTIALLY BY OPIATES AND OPIOID PEPTIDES [J].

CHILDERS, SR ;

CREESE, I ;

SNOWMAN, AM ;

SNYDER, SH .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (01) :11-18

[8]

CREESE I, 1975, J PHARMACOL EXP THER, V194, P205

[9] MULTIPLE OPIATE RECEPTOR-SITES ON PRIMARY AFFERENT-FIBERS [J].

FIELDS, HL ;

EMSON, PC ;

LEIGH, BK ;

GILBERT, RFT ;

IVERSEN, LL .

NATURE, 1980, 284 (5754) :351-353

[10] INHIBITORY POTENCY OF VARIOUS PEPTIDES ON ENKEPHALINASE ACTIVITY FROM MOUSE STRIATUM [J].

FOURNIEZALUSKI, MC ;

PERDRISOT, R ;

GACEL, G ;

SWERTS, JP ;

ROQUES, BP ;

SCHWARTZ, JC .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 91 (01) :130-135

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