STUDIES DIRECTED TOWARD THE TOTAL SYNTHESIS OF THE RUBRADIRIN ANTIBIOTICS .2. SYNTHESIS OF THE UNIQUE MORPHOLINONAPHTHOQUINONE CHROMOPHORE - A LESSON IN DIELS-ALDER REGIOCONTROL BY DIENE SUBSTITUENT SELECTION

被引：13

作者：

KOZIKOWSKI, AP ^{[1
]}

SUGIYAMA, K ^{[1
]}

SPRINGER, JP ^{[1
]}

机构：

[1] MERCK SHARP & DOHME,RES LABS,RAHWAY,NJ 07065

来源：

关键词：

D O I：

10.1021/jo00324a054

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：2426 / 2428

页数：3

共 26 条

[1] DIRECT ALPHA-LITHIATION OF PHENOXYACETIC ACID AND ELECTROPHILIC SUBSTITUTION
ADAM, W
FICK, HH
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (04) : 772 - 773
[2] ADAM W, 1978, SYNTHESIS, V10, P828
[3] BHUYAN B. K., 1965, P91
[4] CASINI G, 1969, FARMACO-ED SCI, V24, P732
[5] REMOVAL OF SULFUR GROUPS FROM MOLECULES BY COPPER(I) - PREPARATION OF SULFUR-SUBSTITUTED 1,3-DIENES FOR DIELS-ALDER REACTION
COHEN, T
MURA, AJ
SHULL, DW
FOGEL, ER
RUFFNER, RJ
FALCK, JR
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1976, 41 (19) : 3218 - 3219
[6] COHEN T, 1980, TETRAHEDRON LETT, P3955
[7] Cohen T., 1979, ORG SYNTH, V59, P202
[8] COREY EJ, 1976, TETRAHEDRON LETT, P809
[9] CHEMISTRY OF RUBRADIRIN .3. RUBRADIRIC ACIDS AND THE STRUCTURE OF RUBRADIRIN
HOEKSEMA, H
MIZSAK, SA
BACZYNSKYJ, L
[J]. JOURNAL OF ANTIBIOTICS, 1979, 32 (07) : 773 - 776
[10] CHEMISTRY OF RUBRADIRINS .1. STRUCTURES OF RUBRANSAROLS-A AND B
HOEKSEMA, H
CHIDESTER, C
MIZSAK, SA
BACZYNSKYJ, L
[J]. JOURNAL OF ANTIBIOTICS, 1978, 31 (10) : 1067 - 1069