OXIDATIVE CYCLIZATIONS WITH PALLADIUM ACETATE - A SHORT SYNTHESIS OF STAUROSPORINE AGLYCONE

被引：87

作者：

HARRIS, W ^{[1
]}

HILL, CH ^{[1
]}

KEECH, E ^{[1
]}

MALSHER, P ^{[1
]}

机构：

[1] ROCHE PROD LTD,RES CTR,WELWYN GARDEN CIT AL7 3AY,HERTS,ENGLAND

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 51期

关键词：

D O I：

10.1016/S0040-4039(00)61431-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A palladium acetate mediated oxidative cyclisation has been used as the key step for the syntheses of staurosporine aglycone and related analogues.

引用

页码：8361 / 8364

页数：4

共 18 条

[1]

AKERMARK B, 1975, J ORG CHEM, V40, P1365, DOI 10.1021/jo00897a048

[2] SYNTHESIS OF INDOLO[2,3-A]PYRROLO[3,4-C]CARBAZOLES BY DOUBLE FISCHER INDOLIZATIONS [J].

BERGMAN, J ;

PELCMAN, B .

JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (04) :824-828

[3]

BIT RA, 1993, IN PRESS TETRAHEDRON

[4] SYNTHESIS OF ARCYRIARUBIN B AND RELATED BISINDOLYLMALEIMIDES [J].

BRENNER, M ;

REXHAUSEN, H ;

STEFFAN, B ;

STEGLICH, W .

TETRAHEDRON, 1988, 44 (10) :2887-2892

[5]

Gill M., 1987, PROG CHEM ORG NAT PR, V51, P216

[6] SYNTHETIC APPROACHES TO INDOLO[2,3-A]CARBAZOLE ALKALOIDS - SYNTHESES OF ARCYRIAFLAVIN-A AND AT2433-B AGLYCONE [J].

GRIBBLE, GW ;

BERTHEL, SJ .

TETRAHEDRON, 1992, 48 (41) :8869-8880

[7] SYNTHESIS OF THE INDOLO[2,3-A]CARBAZOLE NATURAL-PRODUCTS STAUROSPORINONE AND ARCYRIAFLAVIN-B [J].

HUGHES, I ;

NOLAN, WP ;

RAPHAEL, RA .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1990, (09) :2475-2480

[8]

ITAHARA T, 1980, J CHEM SOC CHEM COMM, P49

[9]

ITAHARA T, 1978, SYNTHESIS-STUTTGART, P607

[10] SYNTHESIS OF THE AROMATIC AND MONOSACCHARIDE MOIETIES OF STAUROSPORINE [J].

JOYCE, RP ;

GAINOR, JA ;

WEINREB, SM .

JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (07) :1177-1185

← 1 2 →