SYNTHESIS AND BETA-LACTAMASE INHIBITORY PROPERTIES OF 2-BETA-[(1,2,3-TRIAZOL-1-YL)METHYL]-2-ALPHA-METHYLPENAM-3-ALPHA-CARBOXYLIC ACID 1,1-DIOXIDE AND RELATED TRIAZOLYL DERIVATIVES

被引：112

作者：

MICETICH, RG

MAITI, SN

SPEVAK, P

HALL, TW

YAMABE, S

ISHIDA, N

TANAKA, M

YAMAZAKI, T

NAKAI, A

OGAWA, K

机构：

[1] KOBE COLL RES INST,DIV CHEMOTHERAPY,NISHINOMIYA,JAPAN

[2] TAIHO PHARMACEUT CO LTD,RES INST,TOKUSHIMA,JAPAN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 08期

关键词：

D O I：

10.1021/jm00391a032

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

收藏

页码：1469 / 1474

页数：6

相关论文

共 23 条

[1] ARONOFF S, 1985, 14TH INT C CHEM KYOT
[2] ARONOFF SC, 1984, 24TH INT C ANT AG CH
[3] SUBSTITUTIONS- UND ADDITIONSREAKTIONEN AN SILYLIERTEN ACETYLENEN
BIRKOFER, L
UHLENBRA.H
RITTER, A
[J]. CHEMISCHE BERICHTE-RECUEIL, 1963, 96 (12): : 3280 - &
[4] USE OF TETRABUTYLAMMONIUM AZIDE IN CURTIUS REARRANGEMENT
BRANDSTROM, A
LAMM, B
PALMERTZ, I
[J]. ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1974, B 28 (06): : 699 - 701
[5] CP-45,899, A BETA-LACTAMASE INHIBITOR THAT EXTENDS ANTIBACTERIAL SPECTRUM OF BETA-LACTAMS - INITIAL BACTERIOLOGICAL CHARACTERIZATION
ENGLISH, AR
RETSEMA, JA
GIRARD, AE
LYNCH, JE
BARTH, WE
[J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1978, 14 (03) : 414 - 419
[6] SYNTHESIS AND BETA-LACTAMASE INHIBITORY PROPERTIES OF 2BETA-[(ACYLOXY)METHYL]-2-METHYLPENAM-3ALPHA-CARBOXYLIC ACID 1,1-DIOXIDES
GOTTSTEIN, WJ
HAYNES, UJ
MCGREGOR, DN
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (04) : 518 - 522
[7] SYNTHESIS AND BETA-LACTAMASE INHIBITORY PROPERTIES OF 2-BETA-(CHLOROMETHYL)-2-ALPHA-METHYLPENAM-3-ALPHA-CARBOXYLIC ACID 1,1-DIOXIDE
GOTTSTEIN, WJ
CRAST, LB
GRAHAM, RG
HAYNES, UJ
MCGREGOR, DN
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (12) : 1531 - 1534
[8] MEASUREMENT OF BETA-LACTAMASE ACTIVITY AND RATE OF INACTIVATION OF PENICILLINS BY A PH-STAT ALKALIMETRIC TITRATION METHOD
HOU, JP
POOLE, JW
[J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1972, 61 (10) : 1594 - &
[9] HOWARTH TT, 1976, J CHEM SOC CHEM COMM, P266
[10] ISHIDA N, 1985, 14TH INT C CHEM KYOT