PREPARATION AND BIOLOGICAL EVALUATION OF A POTENTIAL PHOTOAFFINITY LABEL FOR THE PROSTAGLANDIN-H2 THROMBOXANE-A2 RECEPTOR

被引：11

作者：

ARORA, SK

KATTELMAN, EJ

LIM, CT

LEBRETON, GC

VENTON, DL

机构：

[1] UNIV ILLINOIS,DEPT MED CHEM,CHICAGO,IL 60612

[2] UNIV ILLINOIS,DEPT PHARMACOL,CHICAGO,IL 60612

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 05期

关键词：

D O I：

10.1021/jm00388a029

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：918 / 924

页数：7

共 42 条

[1] LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].

ARMSTRONG, RA ;

JONES, RL ;

WILSON, NH .

BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964

[2]

ARORA SK, 1986, 192ND NAT M AM CHEM

[3] IRREVERSIBLE ENZYME INHIBITORS .155. ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF DIHYDROFOLIC REDUCTASE DERIVED FROM 1-[4-(OMEGA-AMINOALKOXY)-3-CHLOROPHENYL]-4,6-DIAMINO-1,2-DIHYDRO-2,2-DIMETHYL-S-TRIAZINES BEARING A TERMINAL SULFONYL FLUORIDE [J].

BAKER, BR ;

JANSON, EE .

JOURNAL OF MEDICINAL CHEMISTRY, 1969, 12 (04) :672-&

[4] SYNTHESIS AND STRUCTURE OF THE PLATELET-AGGREGATION FACTOR THROMBOXANE-A2 [J].

BHAGWAT, SS ;

HAMANN, PR ;

STILL, WC ;

BUNTING, S ;

FITZPATRICK, FA .

NATURE, 1985, 315 (6019) :511-513

[5] AGGREGATION OF BLOOD PLATELETS BY ADENOSINE DIPHOSPHATE AND ITS REVERSAL [J].

BORN, GVR .

NATURE, 1962, 194 (4832) :927-&

[6]

BUNDY G L, 1975, Tetrahedron Letters, V24, P1957

[7] CHARACTERIZATION OF THE PLATELET PROSTAGLANDIN-D2 RECEPTOR - LOSS OF PROSTAGLANDIN-D2 RECEPTORS IN PLATELETS OF PATIENTS WITH MYELOPROLIFERATIVE DISORDERS [J].

COOPER, B ;

AHERN, D .

JOURNAL OF CLINICAL INVESTIGATION, 1979, 64 (02) :586-590

[8] ARYL-2-HALOGENOALKYLAMINES .13. CHLOROETHYLAMINO-DERIVATIVES OF SOME PHENOXYALKANOIC ACIDS AND OF SOME SUBSTITUTED ALPHA-AMINO-ACIDS [J].

DAVIS, W ;

ROBERTS, JJ ;

ROSS, WCJ .

JOURNAL OF THE CHEMICAL SOCIETY, 1955, :890-895

[9] PHOTOAFFINITY LABELS AS PHARMACOLOGICAL TOOLS [J].

FEDAN, JS ;

HOGABOOM, GK ;

ODONNELL, JP .

BIOCHEMICAL PHARMACOLOGY, 1984, 33 (08) :1167-1180

[10] 9,11-EPOXYIMINOPROSTA-5,13-DIENOIC ACID IS A THROMBOXANE-A2 ANTAGONIST IN HUMAN PLATELETS [J].

FITZPATRICK, FA ;

BUNDY, GL ;

GORMAN, RR ;

HONOHAN, T .

NATURE, 1978, 275 (5682) :764-766

← 1 2 3 4 5 →