ACTIONS OF THE BRAIN-PENETRATING H-2-ANTAGONIST ZOLANTIDINE ON HISTAMINE DYNAMICS AND METABOLISM IN RAT-BRAIN

被引:24
作者
HOUGH, LB
JACKOWSKI, S
EBERLE, N
GOGAS, KR
CAMAROTA, NA
CUE, D
机构
关键词
D O I
10.1016/0006-2952(88)90341-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:4707 / 4711
页数:5
相关论文
共 41 条
[1]   AUTO-INHIBITION OF BRAIN HISTAMINE-RELEASE MEDIATED BY A NOVEL CLASS (H-3) OF HISTAMINE-RECEPTOR [J].
ARRANG, JM ;
GARBARG, M ;
SCHWARTZ, JC .
NATURE, 1983, 302 (5911) :832-837
[2]   STEREOSELECTIVITY OF THE HISTAMINE H3-PRESYNAPTIC AUTORECEPTOR [J].
ARRANG, JM ;
SCHWARTZ, JC ;
SCHUNACK, W .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 117 (01) :109-114
[3]   HIGHLY POTENT AND SELECTIVE LIGANDS FOR HISTAMINE RECEPTORS-H-3 [J].
ARRANG, JM ;
GARBARG, M ;
LANCELOT, JC ;
LECOMTE, JM ;
POLLARD, H ;
ROBBA, M ;
SCHUNACK, W ;
SCHWARTZ, JC .
NATURE, 1987, 327 (6118) :117-123
[4]  
AXELROD J, 1970, MOL PHARMACOL, V6, P78
[5]  
BANNON MJ, 1983, PHARMACOL REV, V35, P53
[6]   STRUCTURAL REQUIREMENTS OF IMIDAZOLE COMPOUNDS TO BE INHIBITORS OR ACTIVATORS OF HISTAMINE METHYLTRANSFERASE - INVESTIGATION OF HISTAMINE ANALOGS AND H2-RECEPTOR ANTAGONISTS [J].
BARTH, H ;
LORENZ, W .
AGENTS AND ACTIONS, 1978, 8 (04) :359-365
[7]   MODIFICATION OF ENZYMATIC ISOTOPIC ASSAY OF HISTAMINE AND ITS APPLICATION TO MEASUREMENT OF HISTAMINE IN TISSUES, SERUM AND URINE [J].
BEAVEN, MA ;
HORAKOVA, Z ;
JACOBSEN, S .
CLINICA CHIMICA ACTA, 1972, 37 (NMAR) :91-+
[8]   NEW INHIBITORS OF HISTAMINE-N-METHYLTRANSFERASE [J].
BEAVEN, MA ;
SHAFF, RE .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (02) :183-188
[9]   ZOLANTIDINE (SK-AND-F-95282) IS A POTENT SELECTIVE BRAIN-PENETRATING HISTAMINE H-2-RECEPTOR ANTAGONIST [J].
CALCUTT, CR ;
GANELLIN, CR ;
GRIFFITHS, R ;
LEIGH, BK ;
MAGUIRE, JP ;
MITCHELL, RC ;
MYLEK, ME ;
PARSONS, ME ;
SMITH, IR ;
YOUNG, RC .
BRITISH JOURNAL OF PHARMACOLOGY, 1988, 93 (01) :69-78
[10]  
CROSS SAM, 1977, ACTA PHARMACOL TOX, V41, P116