QUINAZOLINES AND 1,4-BENZODIAZEPINES .77. REACTION OF 2-AMINO-1,4-BENZODIAZEPINES WITH BIFUNCTIONAL ACYLATING AGENTS

被引：20

作者：

FRYER, RI ^{[1
]}

EARLEY, JV ^{[1
]}

BLOUNT, JF ^{[1
]}

机构：

[1] HOFFMANN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1977年 / 42卷 / 13期

关键词：

D O I：

10.1021/jo00433a005

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：2212 / 2219

页数：8

共 12 条

[1] A REARRANGEMENT OF 5-ARYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPINE-2-14-OXIDES [J].

BELL, SC ;

CHILDRESS, SJ .

JOURNAL OF ORGANIC CHEMISTRY, 1962, 27 (05) :1691-&

[2] REARRANGEMENT OF 2-AMINO-5-PHENYL-3H-1,4-BENZODIAZEPINE 4-OXIDES WITH ACETIC ANHYDRIDE [J].

BELL, SC ;

GOCHMAN, C ;

CHILDRESS, SJ .

JOURNAL OF ORGANIC CHEMISTRY, 1963, 28 (11) :3010-&

[3] QUINAZOLINES AND 1,4-BENZODIAZEPINES .39. SYNTHESIS OF DIHYDROIMIDAZO- AND TETRAHYDROPYRIMIDO[1,2-A][1,4]BENZODIAZEPINES [J].

DERIEG, ME ;

FRYER, RI ;

SCHWEINI.RM ;

STERNBAC.LH .

JOURNAL OF MEDICINAL CHEMISTRY, 1968, 11 (04) :912-&

[4] SYNTHETICAL METHODS FOR PREPARATION OF 3-AMINO-2(1H)-QUINOLONES [J].

FRYER, RI ;

STERNBACH, LH ;

BRUST, B .

JOURNAL OF THE CHEMICAL SOCIETY, 1964, (SEP) :3097-&

[5] QUINAZOLINES AND 1,4-BENZODIAZEPINES .22. A REARRANGEMENT OF 5-PHENYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONES [J].

FRYER, RI ;

STERNBACH, LH .

JOURNAL OF ORGANIC CHEMISTRY, 1965, 30 (02) :524-+

[6] A SYNTHESIS OF AMIDINES FROM CYCLIC AMIDES [J].

FRYER, RI ;

EARLEY, JV ;

FIELD, GF ;

ZALLY, W ;

STERNBAC.LH .

JOURNAL OF ORGANIC CHEMISTRY, 1969, 34 (04) :1143-&

[7] ON APPLICATION OF PHASE RELATIONSHIPS TO COMPLEX STRUCTURES .2. GETTING A GOOD START [J].

GERMAIN, G ;

MAIN, P ;

WOOLFSON, MM .

ACTA CRYSTALLOGRAPHICA SECTION B-STRUCTURAL CRYSTALLOGRAPHY AND CRYSTAL CHEMISTRY, 1970, B 26 :274-&

[8]

MAFFRAND JP, 1973, TETRAHEDRON LETT, V36, P3449

[9] QUINAZOLINES AND 1,4-BENZODIAZEPINES .76. REACTIONS OF SOME DI-4-MORPHOLINYLPHOSPHINYLOXY IMINES [J].

NING, RY ;

FRYER, RI ;

MADAN, PB ;

SLUBOSKI, BC .

JOURNAL OF ORGANIC CHEMISTRY, 1976, 41 (16) :2724-2727

[10]

SCHULTE E, 1975, DTSCHE APOTHEKER ZTG, V115, P1253

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