RELATIONSHIP OF AGONIST EFFICACY TO CHANGES IN GABA SENSITIVITY AND ANTICONVULSANT TOLERANCE FOLLOWING CHRONIC BENZODIAZEPINE LIGAND EXPOSURE

被引:53
作者
HERNANDEZ, TD [1 ]
HENINGER, C [1 ]
WILSON, MA [1 ]
GALLAGER, DW [1 ]
机构
[1] YALE UNIV,SCH MED,DEPT PSYCHIAT,ABRAHAM RIBICOFF RES FACIL & CONNECTICUT MENT HLTH CTR,NEW HAVEN,CT 06508
关键词
D O I
10.1016/0014-2999(89)90535-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:145 / 155
页数:11
相关论文
共 28 条
[1]   SINGLE SUBUNITS OF THE GABAA RECEPTOR FORM ION CHANNELS WITH PROPERTIES OF THE NATIVE RECEPTOR [J].
BLAIR, LAC ;
LEVITAN, ES ;
MARSHALL, J ;
DIONNE, VE ;
BARNARD, EA .
SCIENCE, 1988, 242 (4878) :577-579
[2]   LACK OF TOLERANCE OR WITHDRAWAL EFFECTS IN MICE AFTER CHRONIC ADMINISTRATION OF THE NONSEDATING ANXIOLYTIC, CGS-9896 [J].
BOAST, CA ;
GERHARDT, SC .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1987, 26 (03) :601-606
[3]  
FEELY MP, 1988, LANCET, P1460
[4]  
FILE SE, 1987, LANCET, P106
[5]  
FLEISCHHACKER WW, 1988, LANCET, P504
[6]   DEVELOPMENT OF TOLERANCE TO THE ANTICONVULSANT EFFECT OF DIAZEPAM IN DOGS [J].
FREY, HH ;
PHILIPPIN, HP ;
SCHEULER, W .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 104 (1-2) :27-38
[7]   CONTINUOUS RELEASE OF DIAZEPAM - ELECTROPHYSIOLOGICAL, BIOCHEMICAL AND BEHAVIORAL CONSEQUENCES [J].
GALLAGER, DW ;
MALCOLM, AB ;
ANDERSON, SA ;
GONSALVES, SF .
BRAIN RESEARCH, 1985, 342 (01) :26-36
[8]   PERIODIC BENZODIAZEPINE ANTAGONIST ADMINISTRATION PREVENTS BENZODIAZEPINE WITHDRAWAL SYMPTOMS IN PRIMATES [J].
GALLAGER, DW ;
HENINGER, K ;
HENINGER, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 132 (01) :31-38
[9]   ALTERATIONS IN A LOW AFFINITY GABA-RECOGNITION SITE FOLLOWING CHRONIC BENZODIAZEPINE TREATMENT [J].
GALLAGER, DW ;
RAUCH, SL ;
MALCOLM, AB .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 98 (01) :159-160
[10]   CHRONIC BENZODIAZEPINE TREATMENT DECREASES POSTSYNAPTIC GABA SENSITIVITY [J].
GALLAGER, DW ;
LAKOSKI, JM ;
GONSALVES, SF ;
RAUCH, SL .
NATURE, 1984, 308 (5954) :74-77