COMPARISON OF INVITRO POTENCIES IN PHARMACOLOGICAL AND BINDING ASSAYS AFTER INHIBITION OF PEPTIDASES REVEALS THAT DYNORPHIN (1-9) IS A POTENT KAPPA-AGONIST

被引：20

作者：

MCKNIGHT, AT

CORBETT, AD

PATERSON, SJ

MAGNAN, J

KOSTERLITZ, HW

机构：

来源：

LIFE SCIENCES | 1982年 / 31卷 / 16-1期

关键词：

D O I：

10.1016/0024-3205(82)90195-3

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：1725 / 1728

页数：4

共 11 条

[1] DYNORPHIN IS A SPECIFIC ENDOGENOUS LIGAND OF THE KAPPA-OPIOID RECEPTOR [J].

CHAVKIN, C ;

JAMES, IF ;

GOLDSTEIN, A .

SCIENCE, 1982, 215 (4531) :413-415

[2]

CORBETT AD, 1982, NATURE LONDON

[3]

MAGNAN J, 1982, NAUNYNSCHMIEDEBERGS

[4]

MCKNIGHT AT, 1982, EUROP J PHARM

[5]

MINAMINO N, 1981, BIOCHEM BIOPH RES CO, V99, P864, DOI 10.1016/0006-291X(81)91243-2

[6]

OKA T, 1982, EUR J PHARMACOL, V79, P301

[7] RABBIT VAS-DEFERENS - A SPECIFIC BIOASSAY FOR OPIOID KAPPA-RECEPTOR AGONISTS [J].

OKA, T ;

NEGISHI, K ;

SUDA, M ;

MATSUMIYA, T ;

INAZU, T ;

UEKI, M .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 73 (2-3) :235-236

[8] EVIDENCE THAT DYNORPHIN-(1-13) ACTS AS AN AGONIST ON OPIOID K-RECEPTORS [J].

OKA, T ;

NEGISHI, K ;

SUDA, M ;

SAWA, A ;

FUJINO, M ;

WAKIMASU, M .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 77 (2-3) :137-141

[9] A SUBCLASSIFICATION OF KAPPA-SITES IN HUMAN-BRAIN BY USE OF DYNORPHIN 1-17 [J].

PFEIFFER, A ;

PASI, A ;

MEHRAEIN, P ;

HERZ, A .

NEUROPEPTIDES, 1981, 2 (02) :89-97

[10] DYNORPHINS - SIMILAR RELATIVE POTENCIES ON MU-OPIATE, DELTA-OPIATE AND KAPPA-OPIATE RECEPTORS [J].

QUIRION, R ;

PERT, CB .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 76 (04) :467-468

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