S-GLYCOSYLATED CYCLIC-PEPTIDES

被引：36

作者：

GERZ, M ^{[1
]}

MATTER, H ^{[1
]}

KESSLER, H ^{[1
]}

机构：

[1] TECH UNIV MUNICH,INST ORGAN CHEM,LICHTENBERGSTR 4,W-8046 GARCHING,GERMANY

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1993年 / 32卷 / 02期

关键词：

D O I：

10.1002/anie.199302691

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The high chemical and enzymatic stability of thioglycosides stimulated the synthesis of S-glycosylated cyclopeptides. The structural properties of this new class of compounds were established by conformational analysis with 2D NMR methods and molecular dynamics calculations. These substances are of interest for the development of site-specific drugs.

引用

页码：269 / 271

页数：3

共 21 条

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