4-DIAZOCYCLOHEXA-2,5-DIENONES AS PHOTOAFFINITY REAGENTS FOR PROTEINS

被引：13

作者：

KESSLER, P ^{[1
]}

EHRETSABATIER, L ^{[1
]}

GOELDNER, M ^{[1
]}

HIRTH, C ^{[1
]}

机构：

[1] UNIV LOUIS PASTEUR,FAC PHARM,CNRS,URA 1386,CHIM BIOORGAN LAB,BP 24,F-67401 ILLKIRCH GRAFFENS,FRANCE

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 09期

关键词：

D O I：

10.1016/S0040-4039(00)88784-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The protonated 2-(2′-N,N-diethylaminoethyl)-4-diazocyclohexa-2,5-dienone was synthesized and tested as a photoaffinity probe for the active site of acetylcholinesterase, which was efficiently inactivated. © 1990.

引用

页码：1275 / 1278

页数：4

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