3-PHENYL-4-HYDROXYQUINOLIN-2(1H)-ONES - POTENT AND SELECTIVE ANTAGONISTS AT THE STRYCHNINE-INSENSITIVE GLYCINE SITE ON THE N-METHYL-D-ASPARTATE RECEPTOR COMPLEX

被引：83

作者：

MCQUAID, LA ^{[1
]}

SMITH, ECR ^{[1
]}

LODGE, D ^{[1
]}

PRALONG, E ^{[1
]}

WIKEL, JH ^{[1
]}

CALLIGARO, DO ^{[1
]}

OMALLEY, PJ ^{[1
]}

机构：

[1] UNIV LONDON ROYAL VET COLL,LONDON NW1 0TU,ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1992年 / 35卷 / 18期

关键词：

D O I：

10.1021/jm00096a019

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：3423 / 3425

页数：3

共 25 条

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[5] FOSTER AC, 1989, J NEUROSCI, V9, P2191
[6] NOVEL INDOLE-2-CARBOXYLATES AS LIGANDS FOR THE STRYCHNINE-INSENSITIVE N-METHYL-D-ASPARTATE-LINKED GLYCINE RECEPTOR
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[7] Hansch C, 1979, SUBSTITUENT CONSTANT
[8] 4-[(CARBOXYMETHYL)OXY]-5,7-DICHLOROQUINOLINE-2-CARBOXYLIC AND 4-[(CARBOXYMETHYL)AMINO]-5,7-DICHLOROQUINOLINE-2-CARBOXYLIC ACID - NEW ANTAGONISTS OF THE STRYCHNINE-INSENSITIVE GLYCINE BINDING-SITE ON THE N-METHYL-D-ASPARTATE RECEPTOR COMPLEX
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1990, 33 (12) : 3130 - 3132
[9] H-1, F-19 AND C-13 NMR ASSIGNMENTS OF 5,7-DIHALOGENATED KYNURENIC ACID-DERIVATIVES
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[J]. MAGNETIC RESONANCE IN CHEMISTRY, 1991, 29 (08) : 859 - 860
[10] GLYCINE POTENTIATES THE NMDA RESPONSE IN CULTURED MOUSE-BRAIN NEURONS
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[J]. NATURE, 1987, 325 (6104) : 529 - 531

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