2-NITROIMIPRAMINE - A SELECTIVE IRREVERSIBLE INHIBITOR OF [H-3] SEROTONIN UPTAKE AND [H-3] IMIPRAMINE BINDING IN PLATELETS

被引:50
作者
REHAVI, M
ITTAH, Y
RICE, KC
SKOLNICK, P
GOODWIN, FK
PAUL, SM
机构
[1] NIAMDD,CHEM LAB,BETHESDA,MD 20205
[2] NIAMDD,BIOORGAN CHEM LAB,BETHESDA,MD 20205
关键词
D O I
10.1016/0006-291X(81)91255-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:954 / 959
页数:6
相关论文
共 8 条
[1]   HUMAN-PLATELETS POSSESS HIGH-AFFINITY BINDING-SITES FOR H-3-IMIPRAMINE [J].
BRILEY, MS ;
RAISMAN, R ;
LANGER, SZ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 58 (03) :347-348
[2]  
Carlsson A, 1968, J Pharm Pharmacol, V20, P150
[3]   DEMONSTRATION AND EVALUATION OF APPARENT CYTOPLASMIC AND VESICULAR SEROTONIN COMPARTMENTS IN HUMAN PLATELETS [J].
COSTA, JL ;
MURPHY, DL ;
KAFKA, MS .
BIOCHEMICAL PHARMACOLOGY, 1977, 26 (06) :517-521
[4]   HIGH-AFFINITY [IMIPRAMINE-H-3 BINDING IN RAT HYPOTHALAMUS - ASSOCIATION WITH UPTAKE OF SEROTONIN BUT NOT OF NOREPINEPHRINE [J].
LANGER, SZ ;
MORET, C ;
RAISMAN, R ;
DUBOCOVICH, ML ;
BRILEY, M .
SCIENCE, 1980, 210 (4474) :1133-1135
[5]   EFFECT OF IPRONIAZID AND IMIPRAMINE ON THE BLOOD PLATELET 5-HYDROXYTRYPTAMINE LEVEL IN MAN [J].
MARSHALL, EF ;
STIRLING, GS ;
TAIT, AC ;
TODRICK, A .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1960, 15 (01) :35-41
[6]   DEMONSTRATION OF SPECIFIC HIGH-AFFINITY BINDING-SITES FOR (H-3) IMIPRAMINE ON HUMAN-PLATELETS [J].
PAUL, SM ;
REHAVI, M ;
SKOLNICK, P ;
GOODWIN, FK .
LIFE SCIENCES, 1980, 26 (12) :953-959
[7]   SPECIFIC TRICYCLIC ANTI-DEPRESSANT BINDING-SITES IN RAT-BRAIN [J].
RAISMAN, R ;
BRILEY, M ;
LANGER, SZ .
NATURE, 1979, 281 (5727) :148-150
[8]   DEMONSTRATION OF SPECIFIC HIGH-AFFINITY BINDING-SITES FOR [H-3] IMIPRAMINE IN HUMAN-BRAIN [J].
REHAVI, M ;
PAUL, SM ;
SKOLNICK, P ;
GOODWIN, FK .
LIFE SCIENCES, 1980, 26 (26) :2273-2279