PHARMACOLOGICAL REGULATION OF THE PHENCYCLIDINE-BINDING SITE ASSOCIATED WITH THE N-METHYL-D-ASPARTATE RECEPTOR-OPERATED ION CHANNEL

被引:25
作者
JOHNSON, KM [1 ]
SNELL, LD [1 ]
SACAAN, AI [1 ]
JONES, SM [1 ]
机构
[1] UNIV TEXAS,MED BRANCH,DEPT PHARMACOL & TOXICOL,GALVESTON,TX 77550
关键词
D O I
10.1002/ddr.430170405
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:281 / 297
页数:17
相关论文
共 67 条
[1]  
BALSTER RL, 1987, PSYCHOPHARMACOLOGY 3, P1573
[2]  
BALSTER RL, 1988, TRANSDUCTION MECHANI, P122
[3]   A COMPARISON OF PCP-LIKE COMPOUNDS FOR NMDA ANTAGONISM IN 2 INVIVO MODELS [J].
BENNETT, DA ;
BERNARD, PS ;
AMRICK, CL .
LIFE SCIENCES, 1988, 42 (04) :447-454
[4]  
BERRY SC, 1984, BIOCHEM PHARMACOL, V33, P3829, DOI 10.1016/0006-2952(84)90047-9
[5]   THE EFFECT OF THE DIOXOLANES ON AMINO-ACID INDUCED EXCITATION IN THE MAMMALIAN SPINAL-CORD [J].
BERRY, SC ;
ANIS, NA ;
LODGE, D .
BRAIN RESEARCH, 1984, 307 (1-2) :85-90
[6]  
BERRY SC, 1983, EUR J PHARMACOL, P261
[7]   2-METHYL-3,3-DIPHENYL-3-PROPANOLAMINE (2-MDP) SELECTIVELY ANTAGONIZES N-METHYL-ASPARTATE (NMA) [J].
BLAKE, JC ;
DAVIES, SN ;
CHURCH, J ;
MARTIN, D ;
LODGE, D .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1986, 24 (01) :23-25
[8]   BIOCHEMICAL-EVIDENCE THAT GLYCINE ALLOSTERICALLY REGULATES AN NMDA RECEPTOR-COUPLED ION CHANNEL [J].
BONHAUS, DW ;
BURGE, BC ;
MCNAMARA, JO .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 142 (03) :489-490
[9]   DIFFERENCES IN RESULTS FROM INVIVO AND INVITRO STUDIES ON THE USE-DEPENDENCY OF N-METHYLASPARTATE ANTAGONISM BY MK-801 AND OTHER PHENCYCLIDINE RECEPTOR LIGANDS [J].
DAVIES, SN ;
MARTIN, D ;
MILLAR, JD ;
ARAM, JA ;
CHURCH, J ;
LODGE, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 145 (02) :141-151
[10]   PHENCYCLIDINE AND RELATED DRUGS BIND TO THE ACTIVATED N-METHYL-D-ASPARTATE RECEPTOR CHANNEL COMPLEX IN RAT-BRAIN MEMBRANES [J].
FAGG, GE .
NEUROSCIENCE LETTERS, 1987, 76 (02) :221-227