DESIGN AND SYNTHESIS OF PEPTIDE DERIVATIVES OF A 3-DEOXY-D-MANNO-2-OCTULOSONIC ACID (KDO) ANALOG AS NOVEL ANTIBACTERIAL AGENTS ACTING UPON LIPOPOLYSACCHARIDE BIOSYNTHESIS

被引：34

作者：

CLAESSON, A

JANSSON, AM

PRING, BG

HAMMOND, SM

EKSTROM, B

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 12期

关键词：

D O I：

10.1021/jm00395a022

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2309 / 2313

页数：5

共 33 条

[1] PHOSPHONOPEPTIDES, A NEW CLASS OF SYNTHETIC ANTIBACTERIAL AGENTS [J].

ALLEN, JG ;

ATHERTON, FR ;

HALL, MJ ;

HASSALL, CH ;

HOLMES, SW ;

LAMBERT, RW ;

NISBET, LJ ;

RINGROSE, PS .

NATURE, 1978, 272 (5648) :56-58

[2]

ALLEN NE, 1985, ANNU REP MED CHEM, V20, P155

[3] USE OF ESTERS OF N-HYDROXYSUCCINIMIDE IN PEPTIDE SYNTHESIS [J].

ANDERSON, GW ;

CALLAHAN, FM ;

ZIMMERMAN, JE .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1964, 86 (09) :1839-+

[4] SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTIBACTERIAL PHOSPHONOPEPTIDES INCORPORATING (1-AMINOETHYL)PHOSPHONIC ACID AND (AMINOMETHYL)PHOSPHONIC ACID [J].

ATHERTON, FR ;

HASSALL, CH ;

LAMBERT, RW .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (01) :29-40

[5] PEPTIDES OF 2-AMINOPIMELIC ACID - ANTIBACTERIAL AGENTS THAT INHIBIT DIAMINOPIMELIC ACID BIOSYNTHESIS [J].

BERGES, DA ;

DEWOLF, WE ;

DUNN, GL ;

GRAPPEL, SF ;

NEWMAN, DJ ;

TAGGART, JJ ;

GILVARG, C .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (01) :89-95

[6] INHIBITION OF ARABINOSE 5-PHOSPHATE ISOMERASE - AN APPROACH TO THE INHIBITION OF BACTERIAL LIPOPOLYSACCHARIDE BIOSYNTHESIS [J].

BIGHAM, EC ;

GRAGG, CE ;

HALL, WR ;

KELSEY, JE ;

MALLORY, WR ;

RICHARDSON, DC ;

BENEDICT, C ;

RAY, PH .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (06) :717-726

[7] A 2-DEOXY ANALOG OF KDO AS THE 1ST INHIBITOR OF THE ENZYME CMP-KDO SYNTHETASE [J].

CLAESSON, A ;

LUTHMAN, K ;

GUSTAFSSON, K ;

BONDESSON, G .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1987, 143 (03) :1063-1068

[8]

CLAESSON A, IN PRESS J ORG CHEM

[9]

GHALAMBOR MA, 1966, J BIOL CHEM, V241, P3216

[10]

GOLDMAN RC, 1986, J BIOL CHEM, V261, P5831

← 1 2 3 4 →