SYNTHESIS OF 1,4-DIHYDROPYRIDINES UNDER MICROWAVE IRRADIATION

被引：76

作者：

ALAJARIN, R ^{[1
]}

VAQUERO, JJ ^{[1
]}

NAVIO, JLG ^{[1
]}

ALVAREZBUILLA, J ^{[1
]}

机构：

[1] UNIV ALCALA DE HENARES, DEPT QUIM ORGAN, E-28871 ALCALA DE HENARES, SPAIN

来源：

SYNLETT | 1992年 / 04期

关键词：

D O I：

10.1055/s-1992-21345

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A domestic microwave oven has been used to accelerate the Hantzsch synthesis of dialkyl 4-aryl-2,6-dimethyl-1,4-dihydro-3,5-pyridinedicarboxylates 1 and a variant leading to 4,4-dialkyl-2,6-dimethyl-1,4-dihydro-3,5-pyridinedicarbonitriles 2. In comparison with the traditional reflux method, similar or higher yields were obtained.

引用

页码：297 / 298

页数：2

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