CYCLIC ENKEPHALIN ANALOGS CONTAINING ALPHA-AMINO-BETA-MERCAPTO-BETA,BETA-PENTAMETHYLENEPROPIONIC ACID AT POSITION-2 OR POSITION-5

被引：7

作者：

BRYAN, WM

CALLAHAN, JF

CODD, EE

LEMIEUX, C

MOORE, ML

SCHILLER, PW

WALKER, RF

HUFFMAN, WF

机构：

[1] CLIN RES INST MONTREAL, CHEM BIOL & PEPTIDE RES LAB, MONTREAL H2W 1R7, QUEBEC, CANADA

[2] SK&F LABS, DEPT REPROD & DEV TOXICOL, KING OF PRUSSIA, PA 19406 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1989年 / 32卷 / 02期

关键词：

D O I：

10.1021/jm00122a005

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：302 / 304

页数：3

共 28 条

[1]

CHANG KJ, 1979, J BIOL CHEM, V254, P2610

[2] DYNORPHIN IS A SPECIFIC ENDOGENOUS LIGAND OF THE KAPPA-OPIOID RECEPTOR [J].

CHAVKIN, C ;

JAMES, IF ;

GOLDSTEIN, A .

SCIENCE, 1982, 215 (4531) :413-415

[3]

CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099

[4]

CODD EE, 1986, PROG OPIOID RES, V75, P351

[5] SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION INVITRO OF CYCLIC ENKEPHALIN ANALOGS - EFFECT OF CONFORMATIONAL CONSTRAINTS ON OPIATE RECEPTOR SELECTIVITY [J].

DIMAIO, J ;

NGUYEN, TMD ;

LEMIEUX, C ;

SCHILLER, PW .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) :1432-1438

[6] ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].

LORD, JAH ;

WATERFIELD, AA ;

HUGHES, J ;

KOSTERLITZ, HW .

NATURE, 1977, 267 (5611) :495-499

[7]

LORD JAH, 1977, NATURE, V17, P1047

[8] RELATIVE CONFORMATIONAL RIGIDITY IN OXYTOCIN AND [1-PENICILLAMINE]-OXYTOCIN - PROPOSAL FOR RELATIONSHIP OF CONFORMATIONAL FLEXIBILITY TO PEPTIDE HORMONE AGONISM AND ANTAGONISM [J].

MERALDI, JP ;

HRUBY, VJ ;

BREWSTER, AIR .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (04) :1373-1377

[9]

MERALDI JP, 1975, PEPTIDES CHEM STRUCT, P803

[10] SOLID PHASE PEPTIDE SYNTHESIS .1. SYNTHESIS OF A TETRAPEPTIDE [J].

MERRIFIELD, RB .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1963, 85 (14) :2149-&

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