THE ANTAGONISM BY BW-A868C OF PGD2 AND BW245C ACTIVATION OF HUMAN-PLATELET ADENYLATE-CYCLASE

被引:45
作者
TRIST, DG
COLLINS, BA
WOOD, J
KELLY, MG
ROBERTSON, AD
机构
[1] WELLCOME RES LABS,DEPT BIOCHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
[2] WELLCOME RES LABS,DEPT SCI COMP & STAT,BECKENHAM BR3 3BS,KENT,ENGLAND
[3] WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
关键词
D O I
10.1111/j.1476-5381.1989.tb11817.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:301 / 306
页数:6
相关论文
共 15 条
[1]   PROSTAGLANDIN-E RECEPTOR SUBTYPES IN SMOOTH-MUSCLE - AGONIST ACTIVITIES OF STABLE PROSTACYCLIN ANALOGS [J].
DONG, YJ ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 87 (01) :97-107
[2]   THE CLASSIFICATION OF PROSTAGLANDIN DP-RECEPTORS IN PLATELETS AND VASCULATURE USING BW-A868C, A NOVEL, SELECTIVE AND POTENT COMPETITIVE ANTAGONIST [J].
GILES, H ;
LEFF, P ;
BOLOFO, ML ;
KELLY, MG ;
ROBERTSON, AD .
BRITISH JOURNAL OF PHARMACOLOGY, 1989, 96 (02) :291-300
[3]   MODULATION OF HUMAN PLATELET ADENYLATE-CYCLASE BY PROSTACYCLIN (PGX) [J].
GORMAN, RR ;
BUNTING, S ;
MILLER, OV .
PROSTAGLANDINS, 1977, 13 (03) :377-388
[4]   THE USE OF A PROSTACYCLIN ANALOG, [H-3] ILOPROST, FOR STUDYING PROSTACYCLIN-BINDING SITES ON HUMAN-PLATELETS AND NEURONAL HYBRID-CELLS [J].
HALL, JM ;
STRANGE, PG .
BIOSCIENCE REPORTS, 1984, 4 (11) :941-948
[5]   STUDIES ON THE CHARACTERIZATION OF PROSTANOID RECEPTORS - A PROPOSED CLASSIFICATION [J].
KENNEDY, I ;
COLEMAN, RA ;
HUMPHREY, PPA ;
LEVY, GP ;
LUMLEY, P .
PROSTAGLANDINS, 1982, 24 (05) :667-689
[6]   THE USE OF STABLE PROSTAGLANDINS TO INVESTIGATE PROSTACYCLIN (PGI2)-BINDING SITES AND PGI2-SENSITIVE ADENYLATE-CYCLASE IN HUMAN-PLATELET MEMBRANES [J].
LOMBROSO, M ;
NICOSIA, S ;
PAOLETTI, R ;
WHITTLE, BJR ;
MONCADA, S ;
VANE, JR .
PROSTAGLANDINS, 1984, 27 (02) :321-333
[7]  
MILLER OV, 1979, J PHARMACOL EXP THER, V210, P134
[8]  
MILLER OV, 1976, J CYCLIC NUCL PROT, V2, P79
[9]   ENZYME ISOLATED FROM ARTERIES TRANSFORMS PROSTAGLANDIN ENDOPEROXIDES TO AN UNSTABLE SUBSTANCE THAT INHIBITS PLATELET-AGGREGATION [J].
MONCADA, S ;
GRYGLEWSKI, R ;
BUNTING, S ;
VANE, JR .
NATURE, 1976, 263 (5579) :663-665
[10]   HIGHLY SENSITIVE ADENYLATE CYCLASE ASSAY [J].
SALOMON, Y ;
LONDOS, C ;
RODBELL, M .
ANALYTICAL BIOCHEMISTRY, 1974, 58 (02) :541-548