RELEASE OF VASOPRESSIN BY ENKEPHALIN

被引:129
作者
BISSET, GW [1 ]
CHOWDREY, HS [1 ]
FELDBERG, W [1 ]
机构
[1] NATL INST MED RES,LONDON NW3 6RB,ENGLAND
关键词
D O I
10.1111/j.1476-5381.1978.tb08472.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
Leu‐enkephalin, its stable analogue [D‐Ala2‐D‐Leu5]‐enkephalin and the C‐fragment of lipotropin (β endorphin) injected intravenously in the rat produced anti‐diuretic responses which were inhibited reversibly by naloxone. It was shown for Leu‐enkephalin that injection into the cerebral ventricles was at least ten times more effective than intravenous injection and for [D‐Ala2‐D‐Leu5]‐enkephalin that the antidiuretic response was associated with increased excretion of vasopressin in the urine. 1978 British Pharmacological Society
引用
收藏
页码:370 / 371
页数:2
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