BENZODIAZEPINE RECEPTORS STUDIES IN LIVING PRIMATES BY POSITRON EMISSION TOMOGRAPHY - INVERSE AGONIST INTERACTIONS

被引:22
作者
HANTRAYE, P
CHAVOIX, C
GUIBERT, B
FUKUDA, H
BROUILLET, E
DODD, RH
PRENANT, C
CROUZEL, M
NAQUET, R
MAZIERE, M
机构
[1] HOP ORSAY,SERV HOSP FREDERIC JOLIOT,CEA,DEPT BIOL,F-91406 ORSAY,FRANCE
[2] CNRS,DEPT NEUROPHYSIOL APPL,PHYSIOL NERVEUSE LAB,F-91190 GIF SUR YVETTE,FRANCE
[3] CNRS,INST CHIM SUBST NAT,F-91190 GIF SUR YVETTE,FRANCE
关键词
D O I
10.1016/0014-2999(87)90438-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:239 / 247
页数:9
相关论文
共 26 条
  • [1] OPERATIONAL MODELS OF PHARMACOLOGICAL AGONISM
    BLACK, JW
    LEFF, P
    [J]. PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1983, 220 (1219): : 141 - 162
  • [2] BINDING OF [DMCM-H-3, A CONVULSIVE BENZODIAZEPINE LIGAND, TO RAT-BRAIN MEMBRANES - PRELIMINARY STUDIES
    BRAESTRUP, C
    NIELSEN, M
    HONORE, T
    [J]. JOURNAL OF NEUROCHEMISTRY, 1983, 41 (02) : 454 - 465
  • [3] INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS
    BRAESTRUP, C
    SCHMIECHEN, R
    NEEF, G
    NIELSEN, M
    PETERSEN, EN
    [J]. SCIENCE, 1982, 216 (4551) : 1241 - 1243
  • [4] GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS
    BRAESTRUP, C
    NIELSEN, M
    [J]. NATURE, 1981, 294 (5840) : 472 - 474
  • [5] BRAESTRUP C, 1982, PSYCHOPHARMACOL BULL, V18, P8
  • [6] BENZODIAZEPINE RECEPTORS - LABELING IN INTACT ANIMALS WITH [H-3]FLUNITRAZEPAM
    CHANG, RSL
    SNYDER, SH
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (02) : 213 - 218
  • [7] EFFECTS OF 2 CONVULSANT BETA-CARBOLINE DERIVATIVES, DMCM AND BETA-CCM, ON REGIONAL NEUROTRANSMITTER AMINO-ACID LEVELS AND ON INVITRO D-ASPARTATE-H-3 RELEASE IN RODENTS
    CHAPMAN, AG
    CHEETHAM, SC
    HART, GP
    MELDRUM, BS
    WESTERBERG, E
    [J]. JOURNAL OF NEUROCHEMISTRY, 1985, 45 (02) : 370 - 381
  • [8] BEHAVIORAL AND CONVULSANT ACTIONS OF 2 METHYL-ESTERS OF BETA-CARBOLINE-3-CARBOXYLIC ACID IN PHOTOSENSITIVE BABOONS AND IN DBA 2 MICE
    CROUCHER, M
    DESARRO, G
    JENSEN, L
    MELDRUM, B
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 104 (1-2) : 55 - 60
  • [9] CROUCHER MJ, 1983, BRIT J PHARMACOL, V80, pP433
  • [10] CHARACTERIZATION OF CONVULSIONS INDUCED BY METHYL BETA-CARBOLINE-3-CARBOXYLATE IN MICE
    DECARVALHO, LP
    GRECKSCH, G
    CAVALHEIRO, EA
    DODD, RH
    CHAPOUTHIER, G
    ROSSIER, J
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (3-4) : 287 - 293