PREPARATION AND PROPERTIES OF A NEW DALARGINE ANALOG L-TYR-D-ALA-GLY-L-PHE-L-TLE-L-ARG

被引：5

作者：

POSPISEK, J

BESPALOVA, ZD

KOVARIKOVA, E

TITOV, MI

BARTH, T

MEDZIHRADSZKY, K

机构：

[1] HUNGARIAN ACAD SCI, CENT RES INST CHEM, H-1361 BUDAPEST 5, HUNGARY

[2] ACAD MED SCI USSR, CTR CARDIOL, MOSCOW 109801, USSR

来源：

COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS | 1987年 / 52卷 / 07期

关键词：

D O I：

10.1135/cccc19871867

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：1867 / 1871

页数：5

共 12 条

[1] INCREASED ANALGESIC ACTIVITIES OF A FLUORINATED AND A DIMERIC ANALOG OF [D-ALA-2]-METHIONINE ENKEPHALINAMIDE [J].

COY, DH ;

KASTIN, AJ ;

WALKER, MJ ;

MCGIVERN, RF ;

SANDMAN, CA .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1978, 83 (03) :977-983

[2] SYNTHESIS, ENZYMIC DEGRADATION, LIPOPHILIC PROPERTIES, AND BIOLOGICAL-ACTIVITY OF [D-ALANINE2, TERT-BUTYLGLYCINE5]ENKEPHALIN AMIDE [J].

FAUCHERE, JL ;

PETERMANN, C .

HELVETICA CHIMICA ACTA, 1980, 63 (04) :824-831

[3] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY [J].

HUGHES, J ;

SMITH, TW ;

KOSTERLITZ, HW ;

FOTHERGILL, LA ;

MORGAN, BA ;

MORRIS, HR .

NATURE, 1975, 258 (5536) :577-579

[4] ASSESSMENT IN GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN DEPENDENT MONKEY [J].

HUTCHINSON, M ;

KOSTERLITZ, HW ;

LESLIE, FM ;

WATERFIELD, AA ;

TERENIUS, L .

BRITISH JOURNAL OF PHARMACOLOGY, 1975, 55 (04) :541-546

[5] BIOSYNTHESIS OF THE ENKEPHALINS AND ENKEPHALIN-CONTAINING POLYPEPTIDES [J].

LEWIS, RV ;

STERN, AS .

ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1983, 23 :353-372

[6] DOUBLE-ENKEPHALINS - SYNTHESIS, ACTIVITY ON GUINEA-PIG ILEUM, AND ANALGESIC EFFECT [J].

LIPKOWSKI, AW ;

KONECKA, AM ;

SROCZYNSKA, I .

PEPTIDES, 1982, 3 (04) :697-700

[7]

LIPKOWSKI AW, 1983, PEPTIDES 1982, P481

[8]

MEDZIHRADSZKY K, 1983, PEPTIDES 1982, P623

[9]

MEDZIHRADSZKY K, UNPUB

[10] D-ALA2-MET-ENKEPHALINAMIDE - POTENT, LONG-LASTING SYNTHETIC PENTAPEPTIDE ANALGESIC [J].

PERT, CB ;

PERT, A ;

CHANG, JK ;

FONG, BTW .

SCIENCE, 1976, 194 (4262) :330-332

← 1 2 →