INHIBITION OF CYCLIC-AMP PHOSPHODIESTERASE ACTIVITY AND MYOCARDIAL-CONTRACTILITY - EFFECTS OF CILOSTAMIDE, A NOVEL PDE INHIBITOR, AND METHYLISOBUTYLXANTHINE ON RABBIT AND CANINE VENTRICULAR MUSCLE

被引:24
作者
ENDOH, M [1 ]
SATOH, K [1 ]
YAMASHITA, S [1 ]
机构
[1] TOHOKU UNIV, SCH MED, DEPT PHARMACOL, SENDAI, MIYAGI 980, JAPAN
关键词
D O I
10.1016/0014-2999(80)90293-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:43 / 52
页数:10
相关论文
共 21 条
[1]  
ARIENS EJ, 1964, MOL PHARMACOL, V1, P145
[2]   CYCLIC NUCLEOTIDES AND CARDIAC-FUNCTION [J].
DRUMMOND, GI ;
SEVERSON, DL .
CIRCULATION RESEARCH, 1979, 44 (02) :145-153
[3]   ACCUMULATION OF CAMP AND POSITIVE INOTROPIC EFFECT EVOKED BY ISOPROTERENOL UNDER GRADED INHIBITION OF PHOSPHODIESTERASE BY PAPAVERINE IN ISOLATED RABBIT PAPILLARY-MUSCLE [J].
ENDOH, M ;
BRODDE, OE ;
SCHUMANN, HJ .
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 1975, 7 (09) :703-711
[4]   EFFECTS OF PAPAVERINE ON ISOLATED RABBIT PAPILLARY-MUSCLE [J].
ENDOH, M ;
SCHUMANN, HJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1975, 30 (02) :213-220
[5]   EFFECTS OF PAPAVERINE AND ITS INTERACTION WITH ISOPRENALINE AND CARBACHOL ON THE CONTRACTILE-FORCE AND CYCLIC NUCLEOTIDE LEVELS OF THE CANINE VENTRICULAR MYOCARDIUM [J].
ENDOH, M ;
HONMA, M .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 306 (03) :241-248
[6]   ULTRASENSITIVE METHOD FOR SIMULTANEOUS DETERMINATION OF CYCLIC-AMP AND CYCLIC-GMP IN SMALL-VOLUME SAMPLES FROM BLOOD AND TISSUE [J].
HONMA, M ;
SATOH, T ;
TAKEZAWA, J ;
UI, M .
BIOCHEMICAL MEDICINE, 1977, 18 (03) :257-273
[7]  
KOHRI H, 1978, 7TH INT C PHARM PAR, P125
[9]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[10]   DISSOCIATION BETWEEN THE ELECTRO-PHYSIOLOGICAL PROPERTIES AND TOTAL TISSUE CYCLIC GUANOSINE-MONOPHOSPHATE CONTENT OF GUINEA-PIG ATRIA [J].
MIRRO, MJ ;
BAILEY, JC ;
WATANABE, AM .
CIRCULATION RESEARCH, 1979, 45 (02) :225-233