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CRYSTALLOGRAPHIC STUDY OF A BETA-LACTAM INHIBITOR COMPLEX WITH ELASTASE AT 1.84-A RESOLUTION
被引:91
作者
:
NAVIA, MA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
NAVIA, MA
[
1
]
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
SPRINGER, JP
[
1
]
LIN, TY
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
LIN, TY
[
1
]
WILLIAMS, HR
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
WILLIAMS, HR
[
1
]
FIRESTONE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
FIRESTONE, RA
[
1
]
PISANO, JM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
PISANO, JM
[
1
]
DOHERTY, JB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
DOHERTY, JB
[
1
]
FINKE, PE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
FINKE, PE
[
1
]
HOOGSTEEN, K
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
HOOGSTEEN, K
[
1
]
机构
:
[1]
MERCK SHARP & DOHME RES LABS,DEPT MEMBRANE & ARTHRIT RES,RAHWAY,NJ 07065
来源
:
NATURE
|
1987年
/ 327卷
/ 6117期
关键词
:
D O I
:
10.1038/327079a0
中图分类号
:
O [数理科学和化学];
P [天文学、地球科学];
Q [生物科学];
N [自然科学总论];
学科分类号
:
07 ;
0710 ;
09 ;
摘要
:
引用
收藏
页码:79 / 82
页数:4
相关论文
共 27 条
[1]
ELECTRONIC-STRUCTURES OF CEPHALOSPORINS AND PENICILLINS .15. INDUCTIVE EFFECT OF THE 3-POSITION SIDE-CHAIN IN CEPHALOSPORINS
BOYD, DB
论文数:
0
引用数:
0
h-index:
0
BOYD, DB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1984,
27
(01)
: 63
-
66
[2]
BETA-LACTAM NOMENCLATURE
BROWN, AG
论文数:
0
引用数:
0
h-index:
0
BROWN, AG
[J].
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY,
1982,
10
(05)
: 365
-
368
[3]
BUSH BL, 1984, COMPUT CHEM, V8, P1, DOI 10.1016/0097-8485(83)80001-1
[4]
REFINED CRYSTAL-STRUCTURE OF GAMMA-CHYMOTRYPSIN AT 1.9 A RESOLUTION - COMPARISON WITH OTHER PANCREATIC SERINE PROTEASES
COHEN, GH
论文数:
0
引用数:
0
h-index:
0
COHEN, GH
SILVERTON, EW
论文数:
0
引用数:
0
h-index:
0
SILVERTON, EW
DAVIES, DR
论文数:
0
引用数:
0
h-index:
0
DAVIES, DR
[J].
JOURNAL OF MOLECULAR BIOLOGY,
1981,
148
(04)
: 449
-
479
[5]
BETA-LACTAM ANTIBIOTICS - GEOMETRICAL REQUIREMENTS FOR ANTI-BACTERIAL ACTIVITIES
COHEN, NC
论文数:
0
引用数:
0
h-index:
0
COHEN, NC
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1983,
26
(02)
: 259
-
264
[6]
DOHERTY JB, 1986, NATURE, V322, P192, DOI 10.1038/322192a0
[7]
3-DIMENSIONAL MOLECULAR MODELING AND DRUG DESIGN
GUND, P
论文数:
0
引用数:
0
h-index:
0
GUND, P
ANDOSE, JD
论文数:
0
引用数:
0
h-index:
0
ANDOSE, JD
RHODES, JB
论文数:
0
引用数:
0
h-index:
0
RHODES, JB
SMITH, GM
论文数:
0
引用数:
0
h-index:
0
SMITH, GM
[J].
SCIENCE,
1980,
208
(4451)
: 1425
-
1431
[8]
HENDRICKSON WA, 1980, COMPUTING CRYSTALLOG
[9]
STRUCTURES OF PRODUCT AND INHIBITOR COMPLEXES OF STREPTOMYCES-GRISEUS PROTEASE-A AT 1.8 A RESOLUTION - A MODEL FOR SERINE PROTEASE CATALYSIS
JAMES, MNG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
JAMES, MNG
SIELECKI, AR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
SIELECKI, AR
BRAYER, GD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
BRAYER, GD
DELBAERE, LTJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
DELBAERE, LTJ
BAUER, CA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
BAUER, CA
[J].
JOURNAL OF MOLECULAR BIOLOGY,
1980,
144
(01)
: 43
-
88
[10]
JANOFF A, 1985, ANNU REV MED, V36, P207
←
1
2
3
→
共 27 条
[1]
ELECTRONIC-STRUCTURES OF CEPHALOSPORINS AND PENICILLINS .15. INDUCTIVE EFFECT OF THE 3-POSITION SIDE-CHAIN IN CEPHALOSPORINS
BOYD, DB
论文数:
0
引用数:
0
h-index:
0
BOYD, DB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1984,
27
(01)
: 63
-
66
[2]
BETA-LACTAM NOMENCLATURE
BROWN, AG
论文数:
0
引用数:
0
h-index:
0
BROWN, AG
[J].
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY,
1982,
10
(05)
: 365
-
368
[3]
BUSH BL, 1984, COMPUT CHEM, V8, P1, DOI 10.1016/0097-8485(83)80001-1
[4]
REFINED CRYSTAL-STRUCTURE OF GAMMA-CHYMOTRYPSIN AT 1.9 A RESOLUTION - COMPARISON WITH OTHER PANCREATIC SERINE PROTEASES
COHEN, GH
论文数:
0
引用数:
0
h-index:
0
COHEN, GH
SILVERTON, EW
论文数:
0
引用数:
0
h-index:
0
SILVERTON, EW
DAVIES, DR
论文数:
0
引用数:
0
h-index:
0
DAVIES, DR
[J].
JOURNAL OF MOLECULAR BIOLOGY,
1981,
148
(04)
: 449
-
479
[5]
BETA-LACTAM ANTIBIOTICS - GEOMETRICAL REQUIREMENTS FOR ANTI-BACTERIAL ACTIVITIES
COHEN, NC
论文数:
0
引用数:
0
h-index:
0
COHEN, NC
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1983,
26
(02)
: 259
-
264
[6]
DOHERTY JB, 1986, NATURE, V322, P192, DOI 10.1038/322192a0
[7]
3-DIMENSIONAL MOLECULAR MODELING AND DRUG DESIGN
GUND, P
论文数:
0
引用数:
0
h-index:
0
GUND, P
ANDOSE, JD
论文数:
0
引用数:
0
h-index:
0
ANDOSE, JD
RHODES, JB
论文数:
0
引用数:
0
h-index:
0
RHODES, JB
SMITH, GM
论文数:
0
引用数:
0
h-index:
0
SMITH, GM
[J].
SCIENCE,
1980,
208
(4451)
: 1425
-
1431
[8]
HENDRICKSON WA, 1980, COMPUTING CRYSTALLOG
[9]
STRUCTURES OF PRODUCT AND INHIBITOR COMPLEXES OF STREPTOMYCES-GRISEUS PROTEASE-A AT 1.8 A RESOLUTION - A MODEL FOR SERINE PROTEASE CATALYSIS
JAMES, MNG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
JAMES, MNG
SIELECKI, AR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
SIELECKI, AR
BRAYER, GD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
BRAYER, GD
DELBAERE, LTJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
DELBAERE, LTJ
BAUER, CA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
UNIV LUND, DEPT BIOCHEM, S-22007 LUND 7, SWEDEN
BAUER, CA
[J].
JOURNAL OF MOLECULAR BIOLOGY,
1980,
144
(01)
: 43
-
88
[10]
JANOFF A, 1985, ANNU REV MED, V36, P207
←
1
2
3
→