SYNTHESIS AND POTENTIAL ANXIOLYTIC ACTIVITY OF 4-AMINO-PYRIDO[2,3-B]INDOLES

被引：30

作者：

BOLTON, D ^{[1
]}

FORBES, IT ^{[1
]}

HAYWARD, CJ ^{[1
]}

PIPER, DC ^{[1
]}

THOMAS, DR ^{[1
]}

THOMPSON, M ^{[1
]}

UPTON, N ^{[1
]}

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT,HARLOW CM19 5AD,ESSEX,ENGLAND

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1993年 / 3卷 / 10期

关键词：

D O I：

10.1016/S0960-894X(01)80991-4

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A novel series of 4-amino-pyrido[2,3-b]indoles is presented as GABA(A) modulators with good potential as therapeutic agents for the treatment of anxiety disorders.

引用

页码：1941 / 1946

页数：6

共 15 条

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