PHARMACOLOGICAL STUDY OF THE CONTRACTILE ACTIVITY OF LEUKOTRIENE-C4 AND LEUKOTRIENE-D4 ON ISOLATED HUMAN AIRWAY SMOOTH-MUSCLE

被引:142
作者
JONES, TR
DAVIS, C
DANIEL, EE
机构
[1] MCMASTER UNIV,FAC HLTH SCI,DEPT NEUROSCI,HAMILTON L8N 3Z5,ONTARIO,CANADA
[2] MCMASTER UNIV,FAC HLTH SCI,DEPT MED,HAMILTON L8N 3Z5,ONTARIO,CANADA
[3] MERCK FROSST LABS,DEPT PHARMACOL,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA
关键词
D O I
10.1139/y82-087
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:638 / 643
页数:6
相关论文
共 24 条
[1]   SELECTIVE INHIBITOR OF SLOW REACTING SUBSTANCE OF ANAPHYLAXIS [J].
AUGSTEIN, J ;
FARMER, JB ;
LEE, TB ;
SHEARD, P ;
TATTERSALL, ML .
NATURE-NEW BIOLOGY, 1973, 245 (146) :215-217
[2]   ARACHIDONIC-ACID METABOLISM IN POLYMORPHONUCLEAR LEUKOCYTES .5. UNSTABLE INTERMEDIATE IN FORMATION OF DIHYDROXY ACIDS [J].
BORGEAT, P ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (07) :3213-3217
[3]   LEUKOTRIENE-B4 - A MEDIATOR OF VASCULAR-PERMEABILITY [J].
BRAY, MA ;
CUNNINGHAM, FM ;
FORDHUTCHINSON, AW ;
SMITH, MJH .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 72 (03) :483-486
[4]   THE RELEASE OF HISTAMINE AND FORMATION OF A SLOW-REACTING SUBSTANCE (SRS-A) DURING ANAPHYLACTIC SHOCK [J].
BROCKLEHURST, WE .
JOURNAL OF PHYSIOLOGY-LONDON, 1960, 151 (03) :416-435
[5]   STEREOSPECIFIC TOTAL SYNTHESIS OF A SLOW REACTING SUBSTANCE OF ANAPHYLAXIS, LEUKOTRIENE C-1 [J].
COREY, EJ ;
CLARK, DA ;
GOTO, G ;
MARFAT, A ;
MIOSKOWSKI, C ;
SAMUELSSON, B ;
HAMMARSTROM, S .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (04) :1436-1439
[6]   LEUKOTRIENES ARE POTENT CONSTRICTORS OF HUMAN BRONCHI [J].
DAHLEN, SE ;
HEDQVIST, P ;
HAMMARSTROM, S ;
SAMUELSSON, B .
NATURE, 1980, 288 (5790) :484-486
[7]   DIFFERENTIAL EFFECTS OF A PARTIALLY PURIFIED PREPARATION OF SLOW-REACTING SUBSTANCE OF ANAPHYLAXIS ON GUINEA-PIG TRACHEAL SPIRALS AND PARENCHYMAL STRIPS [J].
DRAZEN, JM ;
LEWIS, RA ;
WASSERMAN, SI ;
ORANGE, RP ;
AUSTEN, KF .
JOURNAL OF CLINICAL INVESTIGATION, 1979, 63 (01) :1-5
[8]   COMPARATIVE AIRWAY AND VASCULAR ACTIVITIES OF LEUKOTRIENE-C-1 AND LEUKOTRIENE-D INVIVO AND INVITRO [J].
DRAZEN, JM ;
AUSTEN, KF ;
LEWIS, RA ;
CLARK, DA ;
GOTO, G ;
MARFAT, A ;
COREY, EJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (07) :4354-4358
[9]   LEUKOTRIENE-B, A POTENT CHEMOKINETIC AND AGGREGATING SUBSTANCE RELEASED FROM POLYMORPHONUCLEAR LEUKOCYTES [J].
FORDHUTCHINSON, AW ;
BRAY, MA ;
DOIG, MV ;
SHIPLEY, ME ;
SMITH, MJH .
NATURE, 1980, 286 (5770) :264-265
[10]   RESPONSE OF HUMAN ISOLATED BRONCHIAL AND LUNG PARENCHYMAL STRIPS TO SRS-A AND OTHER MEDIATORS OF ASTHMATIC BRONCHOSPASM [J].
GHELANI, AM ;
HOLROYDE, MC ;
SHEARD, P .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 71 (01) :107-112