PUTATIVE ANXIOLYTICS 8-OH-DPAT, BUSPIRONE AND TVX-Q-7821 ARE AGONISTS AT 5-HT1A AUTORECEPTORS IN THE RAPHE NUCLEI

被引:141
作者
DOURISH, CT [1 ]
HUTSON, PH [1 ]
CURZON, G [1 ]
机构
[1] NATL HOSP,INST NEUROL,DEPT NEUROCHEM,LONDON WC1N 3BG,ENGLAND
关键词
D O I
10.1016/0165-6147(86)90318-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:212 / 214
页数:3
相关论文
共 23 条
[1]   8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN, A NEW CENTRALLY ACTING 5-HYDROXYTRYPTAMINE RECEPTOR AGONIST [J].
ARVIDSSON, LE ;
HACKSELL, U ;
NILSSON, JLG ;
HJORTH, S ;
CARLSSON, A ;
LINDBERG, P ;
SANCHEZ, D ;
WIKSTROM, H .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (08) :921-923
[2]  
CUNNINGHAM K A, 1985, Society for Neuroscience Abstracts, V11, P45
[3]  
DAVIES M, 1985, British Journal of Pharmacology, V86, p594P
[4]   H-3-TVX Q-7821 - IDENTIFICATION OF 5-HT1 BINDING-SITES AS TARGET FOR A NOVEL PUTATIVE ANXIOLYTIC [J].
DOMPERT, WU ;
GLASER, T ;
TRABER, J .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 328 (04) :467-470
[5]   LOW-DOSES OF THE PUTATIVE SEROTONIN AGONIST 8-HYDROXY-2-(DI-N-PROPYLAMINO) TETRALIN (8-OH-DPAT) ELICIT FEEDING IN THE RAT [J].
DOURISH, CT ;
HUTSON, PH ;
CURZON, G .
PSYCHOPHARMACOLOGY, 1985, 86 (1-2) :197-204
[6]  
DOURISH CT, 1986, APPETITE
[7]   ANTICONFLICT EFFECT OF THE PUTATIVE SEROTONIN RECEPTOR AGONIST 8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN (8-OH-DPAT) [J].
ENGEL, JA ;
HJORTH, S ;
SVENSSON, K ;
CARLSSON, A ;
LILJEQUIST, S .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 105 (3-4) :365-368
[8]   BIOCHEMICAL ASSESSMENT OF THE CENTRAL 5-HT AGONIST ACTIVITY OF RU-24969 (A PIPERIDINYL INDOLE) [J].
EUVRARD, C ;
BOISSIER, JR .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 63 (01) :65-72
[9]  
Goldberg H L, 1979, Psychopharmacol Bull, V15, P90
[10]   IDENTIFICATION OF PRE-SYNAPTIC SEROTONIN AUTORECEPTORS USING A NEW LIGAND - H-3-PAT [J].
GOZLAN, H ;
ELMESTIKAWY, S ;
PICHAT, L ;
GLOWINSKI, J ;
HAMON, M .
NATURE, 1983, 305 (5930) :140-142