THE SYNTHESIS OF 1-AMINOBENZYLPHOSPHONIC ACIDS FROM BENZYLIDENEDIPHENYLMETHYLAMINES, FOR USE AS STRUCTURAL UNITS IN ANTITHROMBOTIC TRIPEPTIDES

被引：33

作者：

GREEN, D

PATEL, G

ELGENDY, S

BABAN, JA

CLAESON, G

KAKKAR, VV

DEADMAN, J

机构：

来源：

TETRAHEDRON | 1994年 / 50卷 / 17期

关键词：

D O I：

10.1016/S0040-4020(01)90420-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Acid hydrolyses of 0,0-dimethyl or 0,0-diethyl 1-(diphenylmethylamino) benzylphosphonate intermediates 2, formed from the addition at elevated temperature of dimethyl or diethyl phosphite to benzylidenediphenylmethylamines 1, generates 1-aminobenzylphosphonic acids 3 in good yield.

引用

页码：5099 / 5108

页数：10

共 32 条

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