SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF CERTAIN QUINOLINE DERIVATIVES

被引：10

作者：

ABDALLA, MA

AHMED, AHN

ELZOHRY, MF

OMAR, FA

机构：

[1] ASSIUT UNIV,FAC SCI,DEPT CHEM,ASSIUT 71516,EGYPT

[2] ASSIUT UNIV,FAC PHARM,DEPT PHARMACEUT CHEM,ASSIUT 71516,EGYPT

来源：

COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS | 1992年 / 57卷 / 07期

关键词：

D O I：

10.1135/cccc19921547

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Some aryl or heterocyclic mercaptans reacted with 8-quinolyl chloroacetate II or 8-quinolinoxyacetyl chloride IV to give the corresponding 8-quinolyl-alpha-mercaptoacetate V or 8-quinolyloxy thioacetate VI, respectively. The mercaptans V were oxidized to the corresponding sulfones VII. Some of these compounds were tested for their antimicrobial activities in comparison with tetracycline reference compound.

引用

页码：1547 / 1552

页数：6

共 19 条

[1]

ABDELHADI AZ, 1986, POL J PHARM PHARM, V38, P99

[2]

BEERLEV WN, 1960, ANN TROP MED PARASIT, V62, P288

[3]

BEHERA B., 1967, J INDIAN CHEM SOC, V44, P119

[4]

CHAURASIA M R, 1979, Indian Journal of Pharmaceutical Sciences, V41, P152

[5]

CLAYSON DB, 1967, BIOCHEM PHARMACOL, V16, P614

[6]

Collin C H, 1964, MICROBIOLOGICAL METH, P92

[7]

GHONEIM KM, 1987, EGYPT J PHARM SCI, V28, P17

[8] SOME TRANSITION-METAL CHELATES OF 8-HYDROXYQUINOLINE-5-SULFONAMIDES AS POSSIBLE DRUGS [J].

IBRAHIM, SA ;

MAKHLOUF, MT ;

ABDELHAFEZ, AA ;

MOHARRAM, AM .

JOURNAL OF INORGANIC BIOCHEMISTRY, 1986, 28 (01) :57-65

[9]

KHALIL ZH, 1987, J INDIAN CHEM SOC, V64, P42

[10]

MUELLER WMR, 1979, CHEM BER, V112, P2095

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