IRREVERSIBLE BLOCKADE OF [SPIPERONE-H-3-LABELED BUT NOT [DOPAMINE-H-3-LABELED DOPAMINE-RECEPTORS WITH PHENOXYBENZAMINE

被引:20
作者
TITELER, M
机构
关键词
D O I
10.1016/0006-2952(81)90489-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3031 / 3037
页数:7
相关论文
共 24 条
[1]   CHLOROETHYLNORAPOMORPHINE, A PROPOSED LONG-ACTING DOPAMINE ANTAGONIST - INTERACTIONS WITH DOPAMINE-RECEPTORS OF MAMMALIAN FOREBRAIN INVITRO [J].
BALDESSARINI, RJ ;
KULA, NS ;
ARANA, GW ;
NEUMEYER, JL ;
LAW, SJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 67 (01) :105-110
[2]   DOMPERIDONE-H-3 - SELECTIVE LIGAND FOR DOPAMINE RECEPTORS [J].
BAUDRY, M ;
MARTRES, MP ;
SCHWARTZ, JC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 308 (03) :231-237
[3]  
BURT DR, 1976, MOL PHARMACOL, V12, P800
[4]  
FIELDS JZ, 1977, BRAIN RES, V136, P569
[5]  
FURCHGOTT RF, 1972, HDB EXP PHARM, V33, P382
[6]   HEPATIC ALPHA-ADRENORECEPTOR - SPECIFIC AND IRREVERSIBLE LABELING BY [PHENOXYBENZAMINE-H-3 [J].
GUELLAEN, G ;
HANOUNE, J .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 89 (04) :1178-1185
[7]   PHENOXYBENZAMINE DISCRIMINATES MULTIPLE DOPAMINE-RECEPTORS [J].
HAMBLIN, M ;
CREESE, I .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 65 (01) :119-121
[8]   COMPARISON OF EFFECT OF NEUROLEPTIC DRUGS ON BINDING OF HALOPERIDOL-H-3 AND CIS(Z)-FLUPENTHIXOL-H-3 AND ON ADENYLATE-CYCLASE ACTIVITY IN RAT STRIATAL TISSUE INVITRO [J].
HYTTEL, J .
PROGRESS IN NEURO-PSYCHOPHARMACOLOGY, 1978, 2 (03) :329-335
[9]   DISTINCTION BETWEEN DOPAMINERGIC AND SEROTONERGIC COMPONENTS OF NEUROLEPTIC BINDING-SITES IN LIMBIC BRAIN AREAS [J].
LEYSEN, JE ;
GOMMEREN, W ;
LADURON, PM .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (03) :447-448
[10]   RESOLUTION OF DOPAMINE AND SEROTONIN RECEPTOR COMPONENTS OF [SPIPERONE-H-3 BINDING TO RAT-BRAIN REGIONS [J].
LIST, SJ ;
SEEMAN, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (04) :2620-2624