A SINGLE POINT MUTATION CONFERS TETRODOTOXIN AND SAXITOXIN INSENSITIVITY ON THE SODIUM CHANNEL-II

被引:303
作者
NODA, M
SUZUKI, H
NUMA, S
STUHMER, W
机构
[1] MAX PLANCK INST BIOPHYS CHEM,POSTFACH 2841,W-3400 GOTTINGEN,GERMANY
[2] KYOTO UNIV,FAC MED,DEPT MED CHEM,KYOTO 606,JAPAN
[3] KYOTO UNIV,FAC MED,DEPT MOLEC GENET,KYOTO 606,JAPAN
关键词
D O I
10.1016/0014-5793(89)81531-5
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:213 / 216
页数:4
相关论文
共 31 条
[1]   A RAT-BRAIN NA+ CHANNEL ALPHA-SUBUNIT WITH NOVEL GATING PROPERTIES [J].
AULD, VJ ;
GOLDIN, AL ;
KRAFTE, DS ;
MARSHALL, J ;
DUNN, JM ;
CATTERALL, WA ;
LESTER, HA ;
DAVIDSON, N ;
DUNN, RJ .
NEURON, 1988, 1 (06) :449-461
[2]   CHEMICAL MODIFICATION OF CRAB NERVES CAN MAKE THEM INSENSITIVE TO LOCAL-ANESTHETICS TETRODOTOXIN AND SAXITOXIN [J].
BAKER, PF ;
RUBINSON, KA .
NATURE, 1975, 257 (5525) :412-414
[3]   MOLECULAR-PROPERTIES OF VOLTAGE-SENSITIVE SODIUM-CHANNELS [J].
CATTERALL, WA .
ANNUAL REVIEW OF BIOCHEMISTRY, 1986, 55 :953-985
[4]   MESSENGER-RNA FROM HUMAN-BRAIN INDUCES DRUG-OPERATED AND VOLTAGE-OPERATED CHANNELS IN XENOPUS OOCYTES [J].
GUNDERSEN, CB ;
MILEDI, R ;
PARKER, I .
NATURE, 1984, 308 (5958) :421-424
[5]  
GUY RH, 1988, MOL BIOL IONIC CHANN, V33, P289
[6]  
HENDERSON R, 1974, P NATL ACAD SCI USA, V71, P3936
[7]   RECEPTOR FOR TETRODOTOXIN AND SAXITOXIN - STRUCTURAL HYPOTHESIS [J].
HILLE, B .
BIOPHYSICAL JOURNAL, 1975, 15 (06) :615-619
[8]  
Hille B, 1984, IONIC CHANNELS EXCIT
[9]   COMPARISON OF IONIC SELECTIVITY OF BATRACHOTOXIN-ACTIVATED CHANNELS WITH DIFFERENT TETRODOTOXIN DISSOCIATION-CONSTANTS [J].
HUANG, LYM ;
CATTERALL, WA ;
EHRENSTEIN, G .
JOURNAL OF GENERAL PHYSIOLOGY, 1979, 73 (06) :839-854
[10]   PRIMARY STRUCTURE OF RAT-BRAIN SODIUM CHANNEL-III DEDUCED FROM THE CDNA SEQUENCE [J].
KAYANO, T ;
NODA, M ;
FLOCKERZI, V ;
TAKAHASHI, H ;
NUMA, S .
FEBS LETTERS, 1988, 228 (01) :187-194