CHEMISTRY OF 2H-3,1-BENZOXAZINE-2,4-(1H)DIONE (ISATOIC ANHYDRIDE) .3. ONE-STEP SYNTHESIS OF 2,3-DIHYDRO-4,1,6-BENZOXADIAZONINE-5,7-(1H,6H)DIONES

被引：10

作者：

BARCZA, S

COPPOLA, GM

SHAPIRO, MJ

机构：

[1] Department of Medicinal Chemistry, Pharmaceutical Division, Sandox, Inc, East Hanover, New Jersey, 07936

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1979年 / 16卷 / 03期

关键词：

D O I：

10.1002/jhet.5570160305

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reactions of N‐haloalkylisatoic anhydrides with amines to produce piperidinobenzamides (2), pyrrolidinobenzamides (4 and 5), and 2,3‐dihydro‐6‐methyl‐4,1,6‐benzoxadiazonine‐5,7‐(1H,6H)diones (10) are described. Spectral data are also discussed. Copyright © 1979 Journal of Heterocyclic Chemistry

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页码：439 / 443

页数：5

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