TACHYKININ ANTAGONIST I - SPECIFIC, COMPETITIVE AND TISSUE-SELECTIVE NEUROKININ-B ANTAGONISTS ON CONTRACTILE ACTIVITY IN SMOOTH MUSCLES

被引:8
作者
HASHIMOTO, T
UCHIDA, Y
NAMINOHIRA, S
SAKAI, T
机构
关键词
D O I
10.1254/jjp.45.570
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:570 / 573
页数:4
相关论文
共 11 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]   NOVEL PHARMACOLOGY OF SUBSTANCE-K-BINDING SITES - A 3RD TYPE OF TACHYKININ RECEPTOR [J].
BUCK, SH ;
BURCHER, E ;
SHULTS, CW ;
LOVENBERG, W ;
ODONOHUE, TL .
SCIENCE, 1984, 226 (4677) :987-989
[3]   BIOLOGICAL EVALUATION OF SUBSTANCE-P ANTAGONISTS [J].
FOLKERS, K ;
HAKANSON, R ;
HORIG, J ;
CHENG, XJ ;
LEANDER, S .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (02) :449-456
[4]   NEUROKININ-B ANALOGS SUBSTITUTED WITH GLYCINE [J].
HASHIMOTO, T ;
MORO, T ;
UCHIDA, Y .
BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 1986, 59 (12) :4006-4008
[5]   NEUROMEDIN-K - A NOVEL MAMMALIAN TACHYKININ IDENTIFIED IN PORCINE SPINAL-CORD [J].
KANGAWA, K ;
MINAMINO, N ;
FUKUDA, A ;
MATSUO, H .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 114 (02) :533-540
[6]   NOVEL NEUROPEPTIDES, NEUROKININ-ALPHA AND NEUROKININ-BETA ISOLATED FROM PORCINE SPINAL-CORD [J].
KIMURA, S ;
OKADA, M ;
SUGITA, Y ;
KANAZAWA, I ;
MUNEKATA, E .
PROCEEDINGS OF THE JAPAN ACADEMY SERIES B-PHYSICAL AND BIOLOGICAL SCIENCES, 1983, 59 (04) :101-104
[7]   NEUROKININ-B IS A PREFERRED AGONIST FOR A NEURONAL SUBSTANCE-P RECEPTOR AND ITS ACTION IS ANTAGONIZED BY ENKEPHALIN [J].
LAUFER, R ;
WORMSER, U ;
FRIEDMAN, ZY ;
GILON, C ;
CHOREV, M ;
SELINGER, Z .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (21) :7444-7448
[8]   THE POSSIBLE EXISTENCE OF MULTIPLE RECEPTORS FOR SUBSTANCE-P [J].
LEE, CM ;
IVERSEN, LL ;
HANLEY, MR ;
SANDBERG, BEB .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 318 (04) :281-287
[9]   SUBSTANCE-P ANTAGONISTS SHOWING SOME SELECTIVITY FOR DIFFERENT RECEPTOR TYPES [J].
REGOLI, D ;
MIZRAHI, J ;
DORLEANSJUSTE, P ;
DION, S ;
DRAPEAU, G ;
ESCHER, E .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 109 (01) :121-125
[10]   SYNTHESES AND BIOLOGICAL-ACTIVITIES OF NEUROKININ-B ANALOGS MODIFIED AT POSITION-2, POSITION-3, AND POSITION-6 [J].
UCHIDA, Y ;
OKIMURA, K ;
KUROSAWA, K ;
SAKURA, N ;
HIROSE, K ;
HASHIMOTO, T .
BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 1987, 60 (04) :1561-1563