FUNCTIONAL EVIDENCE FOR A 2ND BINDING-SITE OF NICOTINIC ANTAGONISTS USING PHENCYCLIDINE DERIVATIVES

被引:24
作者
KLOOG, Y
GABRIALEVITZ, A
KALIR, A
BALDERMAN, D
SOKOLOVSKY, M
机构
[1] ISRAEL INST BIOL RES, NESS ZIONA, ISRAEL
[2] TEL AVIV UNIV, SACKLER SCH MED, TEL AVIV, ISRAEL
关键词
D O I
10.1016/0006-2952(79)90456-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:1447 / 1450
页数:4
相关论文
共 15 条
[1]   AMANTADINE - NEUROMUSCULAR BLOCKADE BY SUPPRESSION OF IONIC CONDUCTANCE OF ACETYLCHOLINE-RECEPTOR [J].
ALBUQUERQUE, EX ;
ELDEFRAWI, AT ;
ELDEFRAWI, ME ;
MANSOUR, NA ;
TSAI, MC .
SCIENCE, 1978, 199 (4330) :788-790
[2]  
Bennett M. V. L., 1971, FISH PHYSIOL, V5, P347, DOI DOI 10.1016/S1546-5098(08)60051-5
[3]  
CHANG C. C., 1963, ARCH INTERNATL PHARMACODYN THER, V144, P241
[4]  
CHANGEUX JP, 1975, COLD SPRING HARB SYM, V40, P211
[5]  
DEGUCHI T, 1971, J PHARMACOL EXP THER, V176, P423
[6]   PERHYDROHISTRIONICOTOXIN - POTENTIAL LIGAND FOR ION CONDUCTANCE MODULATOR OF ACETYLCHOLINE-RECEPTOR [J].
ELDEFRAWI, AT ;
ELDEFRAWI, ME ;
ALBUQUERQUE, EX ;
OLIVEIRA, AC ;
MANSOUR, N ;
ADLER, M ;
DALY, JW ;
BROWN, GB ;
BURGERMEISTER, W ;
WITKOP, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (05) :2172-2176
[7]   ACETYLCHOLINE RECEPTORS - NUMBER AND DISTRIBUTION AT NEUROMUSCULAR JUNCTIONS IN RAT DIAPHRAGM [J].
FAMBROUGH, DM ;
HARTZELL, HC .
SCIENCE, 1972, 176 (4031) :189-+
[8]  
KALIR A, 1978, EUR J MED CHEM, V13, P17
[9]  
KALIR A, 1976, 5TH INT S MED CHEM P, P46
[10]  
KATO G, 1976, MOL PHARMACOL, V12, P92