ONE POT AMIDE/PEPTIDE-SYNTHESIS VIA 2 REDOX REACTIONS

被引：15

作者：

GHOSH, SK ^{[1
]}

SINGH, U ^{[1
]}

MAMDAPUR, VR ^{[1
]}

机构：

[1] BHABHA ATOM RES CTR,DIV BIOORGAN,BOMBAY 400085,INDIA

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(00)77720-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new and highly efficient one-pot self-regulated approach to amide/ peptide synthesis has been developed based on two redox reactions using azide as a latent amine component. For the first time, selenophenol, generated in situ has been found to be an effective reducing agent for the conversion of azides to amines.

引用

页码：805 / 808

页数：4

共 24 条

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