APPLICATION OF THE CYANURATE-ISOCYANURATE REARRANGEMENT TO AMINE SYNTHESIS - PREPARATION OF 2-(2-THIENYL)ETHYLAMINE

被引：5

作者：

HARRINGTON, PJ

SANCHEZ, IH

机构：

[1] Syntex Group Technology Center, Boulder

来源：

SYNTHETIC COMMUNICATIONS | 1993年 / 23卷 / 09期

关键词：

D O I：

10.1080/00397919308011217

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

This communication describes a new method for preparation of 2-(2-thienyl)ethylamine, an important pharmaceutical intermediate. The method is based on the 0-to-N migration of an alkyl group via cyanurate-isocyanurate rearrangement.

引用

页码：1307 / 1314

页数：8

共 49 条

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