A NEW SYNTHESIS OF THE POTENT 5-HT1 RECEPTOR LIGAND, 5-CARBOXYAMIDOTRYPTAMINE (5-CT)

被引：7

作者：

AGARWAL, A ^{[1
]}

JALLURI, RK ^{[1
]}

BLANTON, CD ^{[1
]}

TAYLOR, EW ^{[1
]}

机构：

[1] UNIV GEORGIA,COLL PHARM,DEPT MED CHEM,ATHENS,GA 30602

来源：

SYNTHETIC COMMUNICATIONS | 1993年 / 23卷 / 08期

关键词：

D O I：

10.1080/00397919308018587

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A short, convenient and relatively efficient synthesis of 5-CT is developed through a modified Michael reaction. This method represents a new general synthesis for tryptamines with labile indole substituents.

引用

页码：1101 / 1110

页数：10

共 8 条

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