SOLID-PHASE SYNTHESIS OF PHOSPHONOPEPTIDES

被引：21

作者：

CAMPAGNE, JM ^{[1
]}

COSTE, J ^{[1
]}

JOUIN, P ^{[1
]}

机构：

[1] CNRS,INSERM,CTR PHARMACOL ENDOCRINOL,F-34094 MONTPELLIER 5,FRANCE

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 12期

关键词：

D O I：

10.1016/0040-4039(95)00224-Z

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A solid phase synthesis of a phosphonopeptide is described, in which a type 1 aminophosphonate with a free phosphonic acid was coupled just like an amino acid, using BOP as reagent.

引用

页码：2079 / 2082

页数：4

共 12 条

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[4] SYNTHESIS OF MIXED PHOSPHONATE DIESTER ANALOGS OF DIPEPTIDES USING BOP OR PYBOP REAGENTS
CAMPAGNE, JM
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[J]. TETRAHEDRON LETTERS, 1993, 34 (42) : 6743 - 6744
[5] SOLID-PHASE SYNTHESIS OF PHOSPHINIC PEPTIDES
CAMPAGNE, JM
COSTE, J
GUILLOU, L
HEITZ, A
JOUIN, P
[J]. TETRAHEDRON LETTERS, 1993, 34 (26) : 4181 - 4184
[6] SOLID-PHASE SYNTHESIS OF PEPTIDYLPHOSPHONATES
CAMPBELL, DA
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[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1994, 116 (13) : 6039 - 6040
[7] Guo Jincan, 1994, Journal of the American Chemical Society, V116, P6062, DOI 10.1021/ja00093a002
[8] CHARACTERIZATION OF A MONOCLONAL-ANTIBODY PRODUCED IN AN ATTEMPT TO MIMIC THE ACTIVE-SITE OF HIV ASPARTYL PROTEASE USING HAPTENS BASED ON INHIBITOR MODELS
HANIN, V
CAMPAGNE, JM
DOMINICE, C
MANI, JC
DUFOUR, MN
JOUIN, P
PAU, B
[J]. JOURNAL OF IMMUNOLOGICAL METHODS, 1994, 173 (02) : 139 - 147
[9] MERY J, 1992, PEPTIDE RES, V5, P233
[10] MERY J, 1993, INT J PEPT PROT RES, V42, P44

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