N-[(1-BUTYL-4-PIPERIDINYL)METHYL]-3,4-DIHYDRO-2H-[1,3]OXAZINO[3,2-A]INDOLE-10-CARBOXAMIDE HYDROCHLORIDE - THE FIRST POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST AMIDE WITH ORAL ACTIVITY

被引：32

作者：

GASTER, LM

JOINER, GF

KING, FD

WYMAN, PA

SUTTON, JM

BINGHAM, S

ELLIS, ES

SANGER, GJ

WARDLE, KA

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT,DEPT NEUROL,HARLOW CM19 5AW,ESSEX,ENGLAND

[2] UNIV BATH,SCH CHEM,BATH BA2 7AY,AVON,ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1995年 / 38卷 / 24期

关键词：

D O I：

10.1021/jm00024a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：4760 / 4763

页数：4

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