SYNTHESIS OF [C-14] LABELED N-TERT-BUTYL-ALPHA-PHENYLNITRONE - A POTENTIAL SPIN-TRAPPING AGENT

被引：5

作者：

ANGELINI, G ^{[1
]}

CARNEVALETTI, F ^{[1
]}

PICCININI, F ^{[1
]}

机构：

[1] UNIV MILAN,INST PHARMACOL,APPL PHARMACOL SECT,I-20133 MILAN,ITALY

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1992年 / 31卷 / 04期

关键词：

C-14]-N-TERT-BUTYL-ALPHA-PHENYLNITRONE; SPIN-TRAPPING;

D O I：

10.1002/jlcr.2580310404

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

A single step synthesis of the [C-14-ring]-N-tert-butyl-alpha-phenylnitrone (1) starting from the [C-14-ring] benzaldehyde is described. The product is obtained in high yield (90%) with a good level of purity.

引用

页码：289 / 296

页数：8

共 12 条

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