SUPERNORMAL INSULIN - [D-PHEB24]-INSULIN WITH INCREASED AFFINITY FOR INSULIN-RECEPTORS

被引:57
作者
KOBAYASHI, M [1 ]
OHGAKU, S [1 ]
IWASAKI, M [1 ]
MAEGAWA, H [1 ]
SHIGETA, Y [1 ]
INOUYE, K [1 ]
机构
[1] SHIONOGI RES LABS,OSAKA,JAPAN
关键词
D O I
10.1016/0006-291X(82)91708-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:329 / 336
页数:8
相关论文
共 11 条
[1]  
DEMEYTS P, 1978, NATURE, V273, P504
[2]   MONOIODOINSULIN - DEMONSTRATION OF ITS BIOLOGICAL ACTIVITY AND BINDING TO FAT CELLS AND LIVER MEMBRANES [J].
FREYCHET, P ;
ROTH, J ;
NEVILLE, DM .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1971, 43 (02) :400-&
[3]   SEMISYNTHESIS AND PROPERTIES OF SOME INSULIN ANALOGS [J].
INOUYE, K ;
WATANABE, K ;
TOCHINO, Y .
BIOPOLYMERS, 1981, 20 (09) :1845-1858
[4]   SEMISYNTHESIS AND BIOLOGICAL PROPERTIES OF THE [B24-LEUCINE]-ANALOGUES, [B25-LEUCINE]-ANALOGUES AND [B24-LEUCINE, B25-LEUCINE]-ANALOGUES OF HUMAN INSULIN [J].
INOUYE, K ;
WATANABE, K ;
TOCHINO, Y ;
KANAYA, T ;
KOBAYASHI, M ;
SHIGETA, Y .
EXPERIENTIA, 1981, 37 (08) :811-813
[5]   ENZYME-ASSISTED SEMISYNTHESIS OF HUMAN INSULIN [J].
INOUYE, K ;
WATANABE, K ;
MORIHARA, K ;
TOCHINO, Y ;
KANAYA, T ;
EMURA, J ;
SAKAKIBARA, S .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1979, 101 (03) :751-752
[6]   IMPAIRED NEGATIVE COOPERATIVITY OF THE SEMI-SYNTHETIC ANALOGS HUMAN [LEUB24]-INSULIN AND [LEUB25)-INSULIN [J].
KEEFER, LM ;
PIRON, MA ;
DEMEYTS, P ;
GATTNER, HG ;
DIACONESCU, C ;
SAUNDERS, D ;
BRANDENBURG, D .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 100 (03) :1229-1236
[7]   INSULIN BINDING AND GLUCOSE-UPTAKE OF ADIPOCYTES IN RATS ADAPTED TO HYPER-GRAVITATIONAL FORCE [J].
KOBAYASHI, M ;
MONDON, CE ;
OYAMA, J .
AMERICAN JOURNAL OF PHYSIOLOGY, 1980, 238 (04) :E330-E335
[8]   INSULIN, S-SULFONATE A-CHAIN AND S-SULFONATE B-CHAIN RECEPTOR-BINDING TO HUMAN CULTURED LYMPHOCYTES [J].
KOBAYASHI, M ;
MEEK, JC .
DIABETOLOGIA, 1977, 13 (03) :251-255
[9]   RECEPTOR-BINDING REGION OF INSULIN [J].
PULLEN, RA ;
LINDSAY, DG ;
WOOD, SP ;
TICKLE, IJ ;
BLUNDELL, TL ;
WOLLMER, A ;
KRAIL, G ;
BRANDENBURG, D ;
ZAHN, H ;
GLIEMANN, J ;
GAMMELTOFT, S .
NATURE, 1976, 259 (5542) :369-373
[10]   CHICKEN INSULIN - RADIOIMMUNOLOGICAL CHARACTERIZATION AND ENHANCED ACTIVITY IN RAT FAT-CELLS AND LIVER PLASMA-MEMBRANES [J].
SIMON, J ;
FREYCHET, P ;
ROSSELIN, G .
ENDOCRINOLOGY, 1974, 95 (05) :1439-1449