PROTEIN-BINDING AS A PRIMARY DETERMINANT OF THE CLINICAL PHARMACOKINETIC PROPERTIES OF NONSTEROIDAL ANTIINFLAMMATORY DRUGS

被引:194
作者
LIN, JH [1 ]
COCCHETTO, DM [1 ]
DUGGAN, DE [1 ]
机构
[1] GLAXO INC, RES TRIANGLE PK, NC USA
关键词
D O I
10.2165/00003088-198712060-00002
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:402 / 432
页数:31
相关论文
共 233 条
[1]   INVITRO STUDY OF DRUG DISPLACEMENT INTERACTIONS - WARFARIN-SALICYLATE AND WARFARIN-PHENYLBUTAZONE [J].
AARONS, LJ ;
SCHARY, WL ;
ROWLAND, M .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1979, 31 (05) :322-330
[2]   KINETICS OF DRUG DISPLACEMENT INTERACTIONS [J].
AARONS, LJ ;
ROWLAND, M .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1981, 9 (02) :181-190
[3]   POTENTIATION OF ANTICOAGULANT EFFECT OF WARFARIN BY PHENYLBUTAZONE [J].
AGGELER, PM ;
OREILLY, RA ;
LEONG, L ;
KOWITZ, PE .
NEW ENGLAND JOURNAL OF MEDICINE, 1967, 276 (09) :496-&
[4]  
ANDREASEN F, 1973, ACTA PHARMACOL TOX, V32, P417
[5]  
ANTON AH, 1960, J PHARMACOL EXP THER, V129, P282
[6]   PHARMACOKINETICS OF NAPROXEN IN SUBJECTS WITH NORMAL AND IMPAIRED RENAL-FUNCTION [J].
ANTTILA, M ;
HAATAJA, M ;
KASANEN, A .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 18 (03) :263-268
[7]  
AYRES JW, 1977, RES COMMUN CHEM PATH, V17, P583
[8]   INDOMETHACIN IN RHEUMATOID-ARTHRITIS - CLINICAL EFFECTS, PHARMACOKINETICS, AND PLATELET STUDIES IN RESPONDERS AND NONRESPONDERS [J].
BABER, N ;
HALLIDAY, LDC ;
VANDENHEUVEL, WJA ;
WALKER, RW ;
SIBEON, R ;
KEENAN, JP ;
LITTLER, T ;
ORME, MLE .
ANNALS OF THE RHEUMATIC DISEASES, 1979, 38 (02) :128-136
[9]  
BABER N, 1980, BRIT J CLIN PHARMACO, V10, P387
[10]   ALBUMIN METABOLISM IN RHEUMATOID ARTHRITIS [J].
BALLANTYNE, FC ;
FLECK, A ;
DICK, WC .
ANNALS OF THE RHEUMATIC DISEASES, 1971, 30 (03) :265-+