BINDING OF LOOP DIURETICS TO THEIR RENAL RECEPTORS - USE AS A SCREENING MODEL FOR POTENTIAL DIURETIC ACTIVITY

被引:7
作者
GIESENCROUSE, E [1 ]
FANDELEUR, P [1 ]
WELSCH, C [1 ]
ENGLERT, H [1 ]
LANG, HJ [1 ]
SCHMIDT, M [1 ]
IMBS, JL [1 ]
机构
[1] HOECHST AG,PHARMA SYNTHESE,D-6230 FRANKFURT 80,FED REP GER
关键词
D O I
10.1111/j.1472-8206.1988.tb00628.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:145 / 157
页数:13
相关论文
共 27 条
[1]  
BROOKS BA, 1984, RENAL PHYSIOL BIOCH, V7, P304
[2]   EFFECT OF ETHACRYNIC-ACID ON THICK ASCENDING LIMB OF HENLES LOOP [J].
BURG, M ;
GREEN, N .
KIDNEY INTERNATIONAL, 1973, 4 (05) :301-308
[3]  
ELORY JC, 1982, BR J PHARM, V75, P183
[4]  
FORBUSH B, 1983, J BIOL CHEM, V258, P1787
[5]  
GIEBISCH G, 1985, ARZNEIMITTEL-FORSCH, V35, P336
[6]  
GIESENCROUSE E, 1985, J HYPERTENS, V3, pS211
[7]  
GIESENCROUSE EM, 1986, J PHARMACOL-PARIS, V17, P146
[8]   CHARACTERIZATION OF A HIGH-AFFINITY PIRETANIDE RECEPTOR ON KIDNEY MEMBRANES [J].
GIESENCROUSE, EM ;
WELSCH, C ;
IMBS, JL ;
SCHMIDT, M ;
SCHWARTZ, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 114 (01) :23-31
[9]  
GIESENCROUSE EM, 1987, J BIOL CHEM, V262, P17393
[10]   EVIDENCE FOR ELECTRONEUTRAL SODIUM-CHLORIDE CO-TRANSPORT IN THE CORTICAL THICK ASCENDING LIMB OF HENLE LOOP OF RABBIT KIDNEY [J].
GREGER, R ;
SCHLATTER, E ;
LANG, F .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1983, 396 (04) :308-314