N,N-DIALKYLATED LEUCINE ENKEPHALINS AS POTENTIAL DELTA-OPIOID RECEPTOR ANTAGONISTS

被引：16

作者：

LOVETT, JA ^{[1
]}

PORTOGHESE, PS ^{[1
]}

机构：

[1] UNIV MINNESOTA,COLL PHARM,DEPT MED CHEM,MINNEAPOLIS,MN 55455

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 07期

关键词：

D O I：

10.1021/jm00390a005

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1144 / 1149

页数：6

共 33 条

[1] A REINVESTIGATION OF MIXED CARBONIC ANHYDRIDE METHOD OF PEPTIDE SYNTHESIS [J].

ANDERSON, GW ;

ZIMMERMAN, JE ;

CALLAHAN, FM .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1967, 89 (19) :5012-+

[2]

ANWER MK, 1980, SYNTHESIS-STUTTGART, P929

[3] DIVERGENT STRUCTURE ACTIVITY RELATIONSHIPS IN SERIES OF ENKEPHALIN AGONISTS AND COGNATE ANTAGONISTS [J].

BELTON, P ;

COTTON, R ;

GILES, MB ;

GORMLEY, JJ ;

MILLER, L ;

SHAW, JS ;

TIMMS, D ;

WILKINSON, A .

LIFE SCIENCES, 1983, 33 :443-446

[4] A general procedure of the peptide synthesis. [J].

Bergmann, M ;

Zervas, L .

BERICHTE DER DEUTSCHEN CHEMISCHEN GESELLSCHAFT, 1932, 65 (07) :1192-1201

[5] ENKEPHALIN SYNTHESIS OF 2 PENTAPEPTIDES ISOLATED FROM PORCINE BRAIN WITH RECEPTOR-MEDIATED OPIATE AGONIST ACTIVITY [J].

BOWER, JD ;

GUEST, KP ;

MORGAN, BA .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1976, (23) :2488-2492

[6] ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR [J].

COTTON, R ;

GILES, MG ;

MILLER, L ;

SHAW, JS ;

TIMMS, D .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (3-4) :331-332

[7] SYNTHESIS AND BIOLOGICAL EVALUATION OF PHOSPHONAMIDATE PEPTIDE INHIBITORS OF ENKEPHALINASE AND ANGIOTENSIN-CONVERTING ENZYME [J].

ELLIOTT, RL ;

MARKS, N ;

BERG, MJ ;

PORTOGHESE, PS .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (09) :1208-1216

[8]

GILBERT PE, 1976, J PHARMACOL EXP THER, V198, P66

[9]

HAHN EF, 1977, RES COMMUN CHEM PATH, V18, P1

[10] NEW EXAMPLE OF A MORPHINE-SENSITIVE NEURO-EFFECTOR JUNCTION - ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS [J].

HENDERSON, G ;

HUGHES, J ;

KOSTERLITZ, HW .

BRITISH JOURNAL OF PHARMACOLOGY, 1972, 46 (04) :764-766

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