[H-3] CPP, A NEW COMPETITIVE LIGAND FOR NMDA RECEPTORS

被引:101
作者
OLVERMAN, HJ
MONAGHAN, DT
COTMAN, CW
WATKINS, JC
机构
[1] MED SCH BRISTOL,DEPT PHARMACOL,BRISTOL BS8 1TD,AVON,ENGLAND
[2] UNIV EDINBURGH,DEPT PHARMACOL,EDINBURGH EH8 9YL,MIDLOTHIAN,SCOTLAND
[3] UNIV CALIF IRVINE,DEPT PSYCHOBIOL,IRVINE,CA 92717
关键词
D O I
10.1016/0014-2999(86)90533-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:161 / 162
页数:2
相关论文
共 5 条
[1]   CPP, A NEW POTENT AND SELECTIVE NMDA ANTAGONIST - DEPRESSION OF CENTRAL NEURON RESPONSES, AFFINITY FOR [H-3] D-AP5 BINDING-SITES ON BRAIN MEMBRANES AND ANTICONVULSANT ACTIVITY [J].
DAVIES, J ;
EVANS, RH ;
HERRLING, PL ;
JONES, AW ;
OLVERMAN, HJ ;
POOK, P ;
WATKINS, JC .
BRAIN RESEARCH, 1986, 382 (01) :169-173
[2]   SPECIFIC BINDING OF [H-3]-+2-AMINO-7-PHOSPHONO HEPTANOIC ACID TO RAT-BRAIN MEMBRANES INVITRO [J].
FERKANY, JW ;
COYLE, JT .
LIFE SCIENCES, 1983, 33 (13) :1295-1305
[3]   AUTORADIOGRAPHY OF D-2-[H-3]AMINO-5-PHOSPHONOPENTANOATE BINDING-SITES IN RAT-BRAIN [J].
MONAGHAN, DT ;
YAO, D ;
OLVERMAN, HJ ;
WATKINS, JC ;
COTMAN, CW .
NEUROSCIENCE LETTERS, 1984, 52 (03) :253-258
[4]   L-GLUTAMATE H-3 BINDS TO KAINATE-SENSITIVE, NMDA-SENSITIVE AND AMPA-SENSITIVE BINDING-SITES - AN AUTORADIOGRAPHIC ANALYSIS [J].
MONAGHAN, DT ;
YAO, D ;
COTMAN, CW .
BRAIN RESEARCH, 1985, 340 (02) :378-383
[5]   L-GLUTAMATE HAS HIGHER AFFINITY THAN OTHER AMINO-ACIDS FOR [H-3] D-AP5 BINDING-SITES IN RAT-BRAIN MEMBRANES [J].
OLVERMAN, HJ ;
JONES, AW ;
WATKINS, JC .
NATURE, 1984, 307 (5950) :460-462