TOTAL SYNTHESIS OF ANALOGS OF TOPOSTIN-B, A DNA TOPOISOMERASE-I INHIBITOR .1. SYNTHESIS OF FRAGMENTS OF TOPOSTIN-B-1 ANALOGS

被引：9

作者：

NOGUCHI, H ^{[1
]}

AOYAMA, T ^{[1
]}

SHIOIRI, T ^{[1
]}

机构：

[1] NAGOYA CITY UNIV,FAC PHARMACEUT SCI,MIZUHO KU,NAGOYA,AICHI 467,JAPAN

来源：

TETRAHEDRON | 1995年 / 51卷 / 38期

关键词：

D O I：

10.1016/0040-4020(95)00616-G

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of the right and left building blocks, 36 and 5, for the analog 3 of topostin B-1, an inhibitor of mammalian DNA topoisomerase I, has been achieved in a convenient manner.

引用

页码：10531 / 10544

页数：14

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