SYNTHESIS AND ANTI-INFLAMMATORY ACTIVITY OF 6,11-DIHYDRO-11-OXODIBENZO[B,E]THIEPINALKANOIC ACIDS AND RELATED COMPOUNDS

被引：45

作者：

ACKRELL, J

ANTONIO, Y

FRANCO, F

LANDEROS, R

LEON, A

MUCHOWSKI, JM

MADDOX, ML

NELSON, PH

ROOKS, WH

ROSZKOWSKI, AP

WALLACH, MB

机构：

[1] SYNTEX RES CORP,INST BIOL SCI,PALO ALTO,CA 94304

[2] SYNTEX RES CORP,INST ORGAN CHEM,PALO ALTO,CA 94304

[3] SYNTEX RES CORP,INST PHARMACOL & METAB,PALO ALTO,CA 94304

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1978年 / 21卷 / 10期

关键词：

D O I：

10.1021/jm00208a007

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1035 / 1044

页数：10

共 31 条

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[3] DIBENZ[B,E]OXEPINALKANOIC ACIDS AS NONSTEROIDAL ANTIINFLAMMATORY AGENTS .2. DIHYDRO-10-OXOFURO AND "THIENO[3,2-C][1]BENZOXEPIN-8-ACETIC ACIDS [J].

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[5]

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[6] DIBENZTROPONEACETIC AND DIBENZTROPROPIONIC ACIDS - POTENT NEW ANTIINFLAMMATORY AGENTS [J].

DUNN, JP ;

GREEN, DM ;

NELSON, PH ;

ROOKS, WH ;

TOMOLONIS, A ;

UNTCH, KG .

JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (12) :1557-1562

[7] REACTION OF TEREPHTHALIC ACID WITH FORMALDEHYDE IN SULFUR TRIOXIDE MEDIA [J].

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[8]

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[9]

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[10]

JULOU L, 1971, J PHARMACOL-PARIS, V2, P259

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