MUSCARINIC M2 RECEPTORS IN BOVINE TRACHEAL SMOOTH-MUSCLE - DISCREPANCIES BETWEEN BINDING AND FUNCTION

被引:159
作者
ROFFEL, AF [1 ]
ELZINGA, CRS [1 ]
VANAMSTERDAM, RGM [1 ]
DEZEEUW, RA [1 ]
ZAAGSMA, J [1 ]
机构
[1] UNIV GRONINGEN,DEPT ANALYT CHEM & TOXICOL,9713 AW GRONINGEN,NETHERLANDS
关键词
D O I
10.1016/0014-2999(88)90589-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:73 / 82
页数:10
相关论文
共 39 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]   COMPARISON OF AFFINITY CONSTANTS FOR MUSCARINE-SENSITIVE ACETYLCHOLINE RECEPTORS IN GUINEA-PIG ATRIAL PACEMAKER CELLS AT 29 DEGREESC AND IN ILEUM AT 29 DEGREESC AND 37 DEGREESC [J].
BARLOW, RB ;
BERRY, KJ ;
GLENTON, PAM ;
NIKOLAOU, NM ;
SOH, KS .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (04) :613-620
[3]  
BATINK H D, 1987, British Journal of Pharmacology, V90, p81P
[4]   COMPARISON OF MUSCARINIC ACETYLCHOLINE BINDING IN THE URINARY-BLADDER AND SUBMANDIBULAR-GLAND OF THE RABBIT [J].
BATRA, S .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 138 (01) :83-88
[5]   CHARACTERIZATION OF THE MUSCARINIC RECEPTOR SUBTYPE IN ISOLATED GASTRIC FUNDIC CELLS OF THE RABBIT [J].
BAUDIERE, B ;
MONFERINI, E ;
GIRALDO, E ;
LADINSKY, H ;
BALI, JP .
BIOCHEMICAL PHARMACOLOGY, 1987, 36 (18) :2957-2961
[6]  
BERRIE CP, 1983, BRIT J PHARMACOL, V78, pP67
[7]   COMPARISON OF THE AFFINITY CONSTANT OF SOME MUSCARINIC RECEPTOR ANTAGONISTS WITH THEIR DISPLACEMENT OF [H-3] QUINUCLIDINYL BENZILATE BINDING IN ATRIAL AND ILEAL LONGITUDINAL MUSCLE OF THE GUINEA-PIG [J].
CHOO, LK ;
MITCHELSON, FJ .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1985, 37 (09) :656-658
[8]   FAILURE OF GALLAMINE AND PANCURONIUM TO INHIBIT SELECTIVELY (-)-[H-3]QUINUCLIDINYL BENZILATE BINDING IN GUINEA-PIG ATRIA [J].
CHOO, LK ;
LEUNG, E ;
MITCHELSON, F .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1985, 63 (03) :200-208
[9]   INHIBITORY EFFECT OF GALLAMINE ON MUSCARINIC RECEPTORS [J].
CLARK, AL ;
MITCHELSON, F .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (03) :323-331
[10]   BINDING-STUDIES WITH [H-3] CIS-METHYLDIOXOLANE IN DIFFERENT TISSUES - UNDER CERTAIN CONDITIONS [H-3] CIS-METHYLDIOXOLANE LABELS PREFERENTIALLY BUT NOT EXCLUSIVELY AGONIST HIGH-AFFINITY STATES OF MUSCARINIC M2-RECEPTORS [J].
CLOSSE, A ;
BITTIGER, H ;
LANGENEGGER, D ;
WANNER, A .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 335 (04) :372-377